SCHEMBL7718909

SCHEMBL7718909

CC(C)(C)c1ccc(OC(F)(F)F)c(CNN2CCCCC2c2ccccc2)c1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 16/20 0.43
CFTR P13569 2/20 0.39
CYP2D6 P10635 4/20 0.39
KCNH2 Q12809 2/20 0.37
HTR1A P08908 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HRH1 P35367 1/20 0.37
HTR2B P41595 1/20 0.37
SLC6A3 Q01959 1/20 0.37
TMEM97 Q5BJF2 1/20 0.37
SIGMAR1 Q99720 1/20 0.37
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20178136 0.86 TACR1 (0.55) TACR1CFTRCYP2D6
SCHEMBL8706173 0.82 TACR1 (0.40) TACR1CYP2D6KCNH2HTR1AHTR2A
Hydrochloric Acid SCHEMBL9420087 0.82 TACR1 (0.57) TACR1CYP2D6KCNH2HTR1AHTR2A
SCHEMBL8701944 0.81 TACR1 (0.47) TACR1CYP2D6KCNH2HTR1AHTR2A
Hydrochloric Acid SCHEMBL8706570 0.81 TACR1 (0.41) TACR1CYP2D6KCNH2HTR1AHTR2A
SCHEMBL20178205 0.81 TACR1 (0.46) TACR1CFTRCYP2D6KCNH2HTR1A
Hydrochloric Acid SCHEMBL6384500 0.79 TACR1 (0.48) TACR1CYP2D6KCNH2HTR1AHTR2A
Hydrochloric Acid SCHEMBL8682546 0.77 TACR1 (0.42) TACR1CFTRCYP2D6HTR1AHTR2A
Hydrochloric Acid SCHEMBL8681413 0.76 TACR1 (0.43) TACR1CFTRCYP2D6KCNH2HTR1A
Hydrochloric Acid SCHEMBL8610067 0.76 CFTR (0.40) TACR1CFTRCYP2D6HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6376507-B1 NERVE SYSTEM DISORDERS, AMYOTROPIC LATERAL SCLEROSIS PFIZER INC. 2002-04-23 US disclosed