SCHEMBL20178205

SCHEMBL20178205

COc1ccc(C(F)(F)F)cc1CNN1CCCC1c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 12/20 0.46
CYP2D6 P10635 5/20 0.46
CFTR P13569 2/20 0.42
KCNH2 Q12809 1/20 0.41
KDM1A O60341 1/20 0.40
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
HTR1A P08908 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HRH1 P35367 1/20 0.40
HTR2B P41595 1/20 0.40
SLC6A3 Q01959 1/20 0.40
TMEM97 Q5BJF2 1/20 0.40
SIGMAR1 Q99720 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20178136 0.91 TACR1 (0.55) TACR1CYP2D6CFTRKDM1AMAOA
Hydrochloric Acid SCHEMBL9420087 0.82 TACR1 (0.57) TACR1CYP2D6KCNH2HTR1AHTR2A
Hydrochloric Acid SCHEMBL8682546 0.82 TACR1 (0.42) TACR1CYP2D6CFTRKDM1AMAOA
SCHEMBL8328962 0.81 TACR1 (0.53) TACR1CFTRKDM1AMAOAMAOB
SCHEMBL8328961 0.81 TACR1 (0.53) TACR1CFTRKDM1AMAOAMAOB
SCHEMBL7718909 0.81 TACR1 (0.43) TACR1CYP2D6CFTRKCNH2HTR1A
Hydrochloric Acid SCHEMBL8681413 0.80 TACR1 (0.43) TACR1CYP2D6CFTRKCNH2HTR1A
SCHEMBL1626959 0.80 KMT2A (0.53) TACR1KDM1AMAOAMAOB
Hydrochloric Acid SCHEMBL8683252 0.80 TACR1 (0.41) TACR1CYP2D6CFTRHTR1AHTR2A
Hydrochloric Acid SCHEMBL8681023 0.78 CFTR (0.41) TACR1CYP2D6CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9981910-B2 Substituted pyrrolidines and methods of use ABBVIE S.Á.R.L. (LU) 2018-05-29 US disclosed