SCHEMBL20178136

SCHEMBL20178136

COc1ccc(C(C)(C)C)cc1CNN1CCCC1c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 15/20 0.55
CFTR P13569 2/20 0.47
CYP2D6 P10635 2/20 0.45
KDM1A O60341 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20178205 0.91 TACR1 (0.46) TACR1CFTRCYP2D6KDM1AMAOA
SCHEMBL7718909 0.86 TACR1 (0.43) TACR1CFTRCYP2D6
Hydrochloric Acid SCHEMBL8682546 0.85 TACR1 (0.42) TACR1CFTRCYP2D6KDM1AMAOA
SCHEMBL28873991 0.84 TACR1 (0.44) TACR1CFTRCYP2D6
Hydrochloric Acid SCHEMBL8681413 0.83 TACR1 (0.43) TACR1CFTRCYP2D6
Hydrochloric Acid SCHEMBL8683252 0.82 TACR1 (0.41) TACR1CFTRCYP2D6
SCHEMBL8328961 0.82 TACR1 (0.53) TACR1CFTRKDM1AMAOAMAOB
SCHEMBL8328962 0.82 TACR1 (0.53) TACR1CFTRKDM1AMAOAMAOB
Hydrochloric Acid SCHEMBL8681023 0.81 CFTR (0.41) TACR1CFTRCYP2D6
SCHEMBL1626959 0.81 KMT2A (0.53) TACR1KDM1AMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9981910-B2 Substituted pyrrolidines and methods of use ABBVIE S.Á.R.L. (LU) 2018-05-29 US disclosed