SCHEMBL7719693

SCHEMBL7719693

N#Cc1ccc(C(N)=O)c(Cl)n1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 6/20 0.43
KMT2A Q03164 2/20 0.37
ATM Q13315 1/20 0.37
MYC P01106 1/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
PARP1 P09874 6/20 0.35
SOS2 Q07890 1/20 0.35
PARP2 Q9UGN5 2/20 0.34
PARP15 Q460N3 1/20 0.34
PARP10 Q53GL7 1/20 0.34
NNMT P40261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20599509 0.84 SMN1; SMN2 (0.43) CASP1KMT2APDE4APDE4BPDE4C
SCHEMBL20599378 0.82 PDE4A (0.38) KMT2APDE4APDE4BPDE4CPDE4D
SCHEMBL7722575 0.79 NNMT (0.53) MYCPARP1NNMT
SCHEMBL20599383 0.78 HSP90AB1 (0.38) KMT2APDE4APDE4BPDE4CPDE4D
SCHEMBL29574628 0.78 PDE4A (0.44) PDE4APDE4BPDE4CPDE4D
SCHEMBL20599363 0.78 PDE4A (0.44) PDE4APDE4BPDE4CPDE4D
SCHEMBL20619364 0.78 PDE4A (0.34) PDE4APDE4BPDE4CPDE4DSOS2
SCHEMBL893997 0.75 KMT2A (0.42) CASP1KMT2AATMPARP1NNMT
SCHEMBL26808076 0.74 PDE4B (0.37) KMT2APDE4APDE4BPDE4CPDE4D
SCHEMBL20602090 0.74 ALDH1A1 (0.34) KMT2APDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0728744-B1 Process for the preparation of carboxylic acids of nitrogen-containing heterocycles LONZA AG (CH) 2002-04-10 EP disclosed
EP-0627422-B1 Process for the preparation of carboxamides of nitrogen-containing aromatic heterocycles LONZA AG (CH) 1997-04-09 EP disclosed
EP-0728744-A2 Process for the preparation of carboxylic acids of nitrogen-containing heterocycles LONZA A.G. (CH) 1996-08-28 EP disclosed
EP-0627422-A2 Process for the preparation of carboxamides of nitrogen-containing aromatic heterocycles, as well as their use LONZA A.G. (CH) 1994-12-07 EP disclosed