SCHEMBL7720340

SCHEMBL7720340

O=C(O)Cc1cn(OCc2ccc3ccccc3n2)c2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.46
AKR1B1 P15121 2/20 0.46
MCL1 Q07820 2/20 0.44
CYSLTR1 Q9Y271 7/20 0.44
CYSLTR2 Q9NS75 4/20 0.44
FFAR1 O14842 1/20 0.43
CYP1A2 P05177 1/20 0.42
ALOX5 P09917 1/20 0.42
PDE10A Q9Y233 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8543204 0.77 FFAR1 (0.57) GPBAR1AKR1B1MCL1CYSLTR1CYSLTR2
SCHEMBL10436587 0.74 GPBAR1 (0.53) GPBAR1AKR1B1CYSLTR1CYSLTR2FFAR1
SCHEMBL9680639 0.72 CDC25A (0.53) MCL1
SCHEMBL7593150 0.72 GPBAR1 (0.56) GPBAR1AKR1B1CYSLTR1CYSLTR2FFAR1
SCHEMBL140815 0.71 CYP1A2 (0.65) GPBAR1AKR1B1CYSLTR1CYSLTR2FFAR1
SCHEMBL8595609 0.71 CYSLTR1 (0.50) GPBAR1CYSLTR1CYSLTR2CYP1A2PDE10A
SCHEMBL6089876 0.70 GPBAR1 (0.68) GPBAR1AKR1B1CYSLTR1CYSLTR2FFAR1
SCHEMBL9140671 0.70 LTB4R (0.57) AKR1B1MCL1CYSLTR1CYSLTR2FFAR1
SCHEMBL11883719 0.69 MCL1 (0.46) MCL1
SCHEMBL8541189 0.69 AKR1B1 (0.57) GPBAR1AKR1B1CYSLTR1CYSLTR2FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6376528-B1 SYNERGISTIC MIXTURE G. D. SEARLE & CO. 2002-04-23 US disclosed