SCHEMBL7720923

SCHEMBL7720923

O=C(O)CNCCNCCc1ccc(C(=O)O)cc1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.50
CA2 P00918 3/20 0.50
ALDH1A1 P00352 3/20 0.45
RARB P10826 6/20 0.44
ADRB1 P08588 2/20 0.43
ADRB3 P13945 2/20 0.43
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.41
RARA P10276 1/20 0.41
MAPT P10636 1/20 0.41
MTOR P42345 1/20 0.41
TP53 P04637 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31688904 0.96 CA1 (0.49) CA1CA2ALDH1A1RARBADRB1
SCHEMBL7716598 0.90 S1PR1 (0.48) CA1CA2ALDH1A1RARBADRB1
SCHEMBL31688891 0.86 RARB (0.51) ALDH1A1RARBKMT2AMEN1RARA
SCHEMBL7723455 0.84 ALDH1A1 (0.59) CA1CA2ALDH1A1KMT2AMEN1
SCHEMBL28066274 0.84 SIGMAR1 (0.57) CA1CA2ALDH1A1LMNAHTT
SCHEMBL7721622 0.83 ALDH1A1 (0.57) CA1CA2ALDH1A1KMT2AMEN1
SCHEMBL31688715 0.80 ALDH1A1 (0.52) CA1CA2ALDH1A1ADRB1ADRB3
SCHEMBL288827 0.80 KDM4E (0.55) CA1CA2
SCHEMBL157742 0.80 KEAP1 (0.59) CA2ALDH1A1MAPT
SCHEMBL4233315 0.79 ALDH1A1 (0.57) ALDH1A1RARBADRB1ADRB3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6417396-B1 BY-PRODUCT INHIBITION; REACTING ORGANIC ALKALI OR ALKALINE EARTH METAL CARBOXYLATE, PHOSPHONATE, OR SULFONATE; ACYLATION, PHOSPHORYLATION, SULFONATION, AMIDATION, ALKYLATION, CYCLIZATION, OR CONDENSATION Lambert, Warner 2002-07-09 US disclosed
US-6395930-B1 AMINE SULFIDE PHOSPHATE OR SULFATE REAGENTS WARNER LAMBERT 2002-05-28 US disclosed
US-6121488-A Quenching reagents for solution phase synthesis WARNER-LAMBERT COMPANY (US) 2000-09-19 US disclosed