SCHEMBL7721904

SCHEMBL7721904

CC(C)(C)OC(=O)NCC(=O)NC1C[C@@H](C(=O)Nc2nc3cc(Cl)ccc3o2)N(C(=O)OC(C)(C)C)C1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ANO1 Q5XXA6 1/20 0.41
USP30 Q70CQ3 1/20 0.41
PTGES O14684 11/20 0.40
CYP1A2 P05177 1/20 0.38
POLB P06746 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
NPY5R Q15761 1/20 0.38
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38
ABL1 P00519 1/20 0.37
BCR P11274 1/20 0.37
ALDH1A1 P00352 1/20 0.37
FFAR2 O15552 1/20 0.37
PTGS2 P35354 2/20 0.37
EGFR P00533 1/20 0.35
BTK Q06187 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7728188 0.82 POLB (0.47) CYP1A2POLBCYP3A4CYP2C19CTSL
SCHEMBL7721906 0.77 USP30 (0.39) ANO1USP30PTGESCYP1A2POLB
SCHEMBL24998171 0.77 PTGES (0.48) ANO1USP30PTGESNPY5RFFAR2
SCHEMBL16238597 0.76 ALDH1A1 (0.53) USP30PTGESPOLBNPY5RALDH1A1
SCHEMBL13257793 0.76 ALDH1A1 (0.53) USP30PTGESPOLBNPY5RALDH1A1
SCHEMBL7729234 0.76 HDAC4 (0.44) CYP1A2POLBCYP3A4CYP2C19
SCHEMBL7725703 0.75 POLB (0.43) CYP1A2POLBCYP3A4CYP2C19ABL1
SCHEMBL7731723 0.74 HDAC8 (0.44) CYP1A2POLBCYP3A4CYP2C19
SCHEMBL7734064 0.73 RAB9A (0.47) ALDH1A1
SCHEMBL7726519 0.73 POLB (0.42) USP30CYP1A2POLBCYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6399629-B1 PYRROLIDINES AND PIPERIDINES FOR TREATING MICROBIAL INFECTIONS BY REDUCING EXPORT OF COADMINISTERED ANTIMICROBIAL AGENT OR COMPOUND SYNTHESIZED BY MICROBES FOR THEIR GROWTH; REDUCING IN VIVO AVAILABILITY MICROCIDE PHARMACEUTICALS, INC. 2002-06-04 US disclosed
WO-2000001714-A1 EFFLUX PUMP INHIBITORS MICROCIDE PHARMACEUTICALS, INC. (US) 2000-01-13 WO disclosed