SCHEMBL7721946

SCHEMBL7721946

CC(C)(C)OC(=O)NC[C@H](O)C(=O)N[C@@H]1C[C@@H](C(=O)Nc2ccc(Oc3ccccc3)cc2)N(C(=O)OC(C)(C)C)C1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 4/20 0.41
NPC1 O15118 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
HTRA1 Q92743 1/20 0.39
GHSR Q92847 1/20 0.39
POLB P06746 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
MCL1 Q07820 4/20 0.38
PABPC1 P11940 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPK1 P28482 1/20 0.38
HTT P42858 1/20 0.38
RECQL P46063 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CFTR P13569 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7731475 0.87 HDAC8 (0.44) HDAC8NPC1MEN1KMT2AGHSR
SCHEMBL7721949 0.84 HDAC8 (0.38) HDAC8NPC1MEN1KMT2AHTRA1
SCHEMBL7722273 0.81 NAMPT (0.47) HDAC8NPC1MEN1KMT2AGHSR
SCHEMBL7722271 0.81 NAMPT (0.47) HDAC8NPC1MEN1KMT2AGHSR
SCHEMBL7728341 0.81 BTK (0.38) MEN1KMT2AHTRA1POLBCYP1A2
SCHEMBL7728349 0.81 BTK (0.38) MEN1KMT2AHTRA1POLBCYP1A2
SCHEMBL7727553 0.81 BTK (0.38) MEN1KMT2AHTRA1POLBCYP1A2
SCHEMBL7729067 0.81 BTK (0.38) MEN1KMT2AHTRA1POLBCYP1A2
SCHEMBL7731723 0.78 HDAC8 (0.44) HDAC8NPC1MEN1KMT2AHTRA1
SCHEMBL7727758 0.78 MMP2 (0.36) POLBCYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6399629-B1 PYRROLIDINES AND PIPERIDINES FOR TREATING MICROBIAL INFECTIONS BY REDUCING EXPORT OF COADMINISTERED ANTIMICROBIAL AGENT OR COMPOUND SYNTHESIZED BY MICROBES FOR THEIR GROWTH; REDUCING IN VIVO AVAILABILITY MICROCIDE PHARMACEUTICALS, INC. 2002-06-04 US disclosed