SCHEMBL7731475

SCHEMBL7731475

CC(C)(C)OC(=O)NCC(=O)NC1C[C@@H](C(=O)Nc2ccc(Oc3ccccc3)cc2)N(C(=O)OC(C)(C)C)C1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 6/20 0.44
NPC1 O15118 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
POLB P06746 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
MMP2 P08253 1/20 0.40
MMP9 P14780 1/20 0.40
PABPC1 P11940 1/20 0.40
EPHX2 P34913 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPK1 P28482 1/20 0.40
HTT P42858 1/20 0.40
RECQL P46063 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CFTR P13569 1/20 0.39
GHSR Q92847 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7731723 0.91 HDAC8 (0.44) HDAC8NPC1MEN1KMT2APOLB
SCHEMBL7727250 0.90 LTA4H (0.45) HDAC8NPC1POLBALDH1A1SMN1; SMN2
SCHEMBL7726519 0.90 POLB (0.42) HDAC8NPC1MEN1KMT2APOLB
SCHEMBL7725703 0.88 POLB (0.43) HDAC8NPC1MEN1KMT2APOLB
SCHEMBL7728188 0.88 POLB (0.47) HDAC8NPC1MEN1KMT2APOLB
SCHEMBL7721946 0.87 HDAC8 (0.41) HDAC8NPC1MEN1KMT2APOLB
SCHEMBL7728407 0.86 MEN1 (0.39) HDAC8NPC1MEN1KMT2APOLB
SCHEMBL7728411 0.86 MEN1 (0.39) HDAC8NPC1MEN1KMT2APOLB
SCHEMBL7722104 0.85 PABPC1 (0.45) HDAC8KMT2APOLBCYP1A2CYP3A4
SCHEMBL7728829 0.85 SIRT2 (0.48) HDAC8POLBGHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6399629-B1 PYRROLIDINES AND PIPERIDINES FOR TREATING MICROBIAL INFECTIONS BY REDUCING EXPORT OF COADMINISTERED ANTIMICROBIAL AGENT OR COMPOUND SYNTHESIZED BY MICROBES FOR THEIR GROWTH; REDUCING IN VIVO AVAILABILITY MICROCIDE PHARMACEUTICALS, INC. 2002-06-04 US disclosed