SCHEMBL7721990

SCHEMBL7721990

CCOC(=O)C(F)(F)C(F)(F)C(F)(F)C(=O)Cl.O=C(Cl)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Cl

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
PKM P14618 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
CYP4F2 P78329 2/20 0.33
CYP4A11 Q02928 2/20 0.33
HDAC4 P56524 2/20 0.33
HDAC6 Q9UBN7 2/20 0.33
THRB P10828 1/20 0.33
LMNA P02545 1/20 0.33
HSD17B10 Q99714 1/20 0.33
POLB P06746 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
ABCB11 O95342 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
TSHR P16473 1/20 0.33
HTR2A P28223 1/20 0.33
PMP22 Q01453 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6618678 0.98 ALDH1A1 (0.36) ALDH1A1PKMKDM4EMEN1KMT2A
SCHEMBL27186828 0.88 ALDH1A1 (0.43) ALDH1A1PKMKDM4EMEN1KMT2A
SCHEMBL4007477 0.88 ALDH1A1 (0.43) ALDH1A1PKMKDM4EMEN1KMT2A
SCHEMBL8166839 0.86 ALDH1A1 (0.42) ALDH1A1PKMKDM4EMEN1KMT2A
SCHEMBL8165793 0.86 ALDH1A1 (0.42) ALDH1A1PKMKDM4EMEN1KMT2A
SCHEMBL2050077 0.82 CA1 (0.43) ALDH1A1PKMKDM4EMEN1KMT2A
SCHEMBL3861059 0.80 THRB (0.46) ALDH1A1PKMKDM4EMEN1KMT2A
SCHEMBL5704701 0.80 THRB (0.46) ALDH1A1PKMKDM4EMEN1KMT2A
SCHEMBL197278 0.80 THRB (0.46) ALDH1A1PKMKDM4EMEN1KMT2A
SCHEMBL5704769 0.80 THRB (0.46) ALDH1A1PKMKDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015479-A4 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC MACROCYCLES AND PROCESSES THEREFOR LILLY CO ELI (US) 2002-07-24 EP disclosed
EP-1015479-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC MACROCYCLES AND PROCESSES THEREFOR ELI LILLY AND COMPANY (US) 2000-07-05 EP disclosed
WO-1998057173-A1 COMBINATORIAL PROCESS FOR PREPARING SUBSTITUTED PHENYLALANINE LIBRARIES ELI LILLY AND COMPANY (US) 1998-12-17 WO disclosed
WO-1998046631-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC MACROCYCLES AND PROCESSES THEREFOR ELI LILLY AND COMPANY (US) 1998-10-22 WO disclosed
WO-1998008839-A1 COMBINATORIAL PROCESS FOR PREPARING SUBSTITUTED THIOPHENE LIBRARIES ELI LILLY AND COMPANY (US) 1998-03-05 WO disclosed