SCHEMBL7722975

SCHEMBL7722975

CCc1c(N2CCNCC2)ccc2c1C(=O)NC2=O

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.43
HTR2A P28223 2/20 0.43
DRD2 P14416 2/20 0.43
DRD4 P21917 2/20 0.43
DRD3 P35462 2/20 0.43
HTR2C P28335 1/20 0.43
HTR7 P34969 7/20 0.39
HTR6 P50406 3/20 0.38
HTR5A P47898 1/20 0.38
ADRB1 P08588 1/20 0.36
ALK Q9UM73 1/20 0.36
PIM1 P11309 1/20 0.35
PIM3 Q86V86 1/20 0.35
PIM2 Q9P1W9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7882760 0.99 HTR1A (0.42) HTR1AHTR2ADRD2DRD4DRD3
SCHEMBL5996608 0.89 PARP1 (0.39)
Hydrochloric Acid SCHEMBL7723748 0.87 PARP1 (0.38)
SCHEMBL4552739 0.83 PIM1 (0.36) HTR1AHTR2ADRD2DRD4DRD3
SCHEMBL7883990 0.81 HTR1A (0.38) HTR1AHTR2ADRD2DRD4DRD3
Alcohol SCHEMBL28156339 0.77 HTR7 (0.52) HTR1AHTR2ADRD2DRD4DRD3
SCHEMBL7964016 0.77 KMT2A (0.36)
Hydrochloric Acid SCHEMBL7727011 0.75 KDM4E (0.43)
SCHEMBL8352376 0.75 PARP1 (0.41) HTR2A
SCHEMBL10911536 0.72 GSK3B (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE37729-E1 4-Heteroaryl-1-piperidinealkylamines and derivatives thereof and their therapeutic utility AVENTIS PHARMACEUTICALS INC. 2002-06-04 US disclosed
US-RE37478-E1 COMPOUNDS WITH HETEROCYCLIC AMINO COMPOUNDS AVENTIS PHARMACEUTICALS, INC. 2001-12-18 US disclosed
US-6207680-B1 FOR THERAPY OF PSYCHOLOGICAL DISORDERS AND PAIN AVENTIS PHARMACEUTICALS INC. 2001-03-27 US disclosed
US-RE37029-E1 ANTIPSYCHOTIC AND ANALGESIC AGENTS AVENTIS PHARMACEUTICALS INC. 2001-01-23 US disclosed