SCHEMBL7723009

SCHEMBL7723009

CCC[C@@H](N)c1nc(C(=O)Nc2cnc3cccc(C(C)(C)C)c3c2)co1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 13/20 0.38
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
KDR P35968 2/20 0.35
MAPT P10636 2/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MEN1 O00255 1/20 0.34
ABCB1 P08183 1/20 0.34
HTT P42858 1/20 0.34
KMT2A Q03164 1/20 0.34
ABCG2 Q9UNQ0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7735550 0.84 TRPV1 (0.52) TRPV1NPC1RAB9AALDH1A1KDM4E
SCHEMBL7732568 0.82 TRPV1 (0.40) TRPV1NPC1RAB9AALDH1A1KDM4E
SCHEMBL7732103 0.73 RAB9A (0.53) TRPV1NPC1RAB9AALDH1A1KDM4E
SCHEMBL7732373 0.71 TRPV1 (0.50) TRPV1NPC1RAB9AALDH1A1KDM4E
Trifluoroacetic Acid SCHEMBL7735917 0.71 RAB9A (0.48) TRPV1NPC1RAB9AALDH1A1KDM4E
SCHEMBL7732431 0.71 TRPV1 (0.41) TRPV1NPC1RAB9AMAPTNFKB1
SCHEMBL7733560 0.71 TRPV1 (0.41) TRPV1NPC1RAB9AMAPTNFKB1
SCHEMBL7850751 0.71 TRPV1 (0.44) TRPV1NPC1RAB9AALDH1A1KDM4E
SCHEMBL7734013 0.71 NPC1 (0.45) TRPV1NPC1RAB9AALDH1A1KDM4E
SCHEMBL7733996 0.71 NPC1 (0.50) TRPV1NPC1RAB9AALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436980-B1 TRANSPORT PROTEIN SUPPRESSORS; MICROBIOCIDES ESSENTIAL THERAPEUTICS, INC. 2002-08-20 US disclosed
US-6204279-B1 SECONDARY AMIDE CONTAINING BENZOXAZOLE DERIVATIVES MICROCIDE PHARMACEUTICALS, INC. 2001-03-20 US disclosed
WO-1999037667-A1 EFFLUX PUMP INHIBITORS MICROCIDE PHARMACEUTICALS, INC. (US) 1999-07-29 WO disclosed