SCHEMBL7724583

SCHEMBL7724583

O=C1N=c2cccc(O)c2=N1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DBH P09172 3/20 0.37
MAOA P21397 2/20 0.35
ALDH1A1 P00352 7/20 0.35
ALOX15 P16050 6/20 0.35
HSD17B10 Q99714 6/20 0.35
TDP1 Q9NUW8 6/20 0.35
HPGD P15428 6/20 0.35
CA2 P00918 5/20 0.35
LMNA P02545 4/20 0.35
CA1 P00915 4/20 0.35
RECQL P46063 3/20 0.35
MMP2 P08253 2/20 0.35
EGFR P00533 2/20 0.35
FYN P06241 2/20 0.35
MMP9 P14780 2/20 0.35
CDK2 P24941 2/20 0.35
ADAMTS4 O75173 1/20 0.35
MMP8 P22894 1/20 0.35
CA6 P23280 1/20 0.35
MMP12 P39900 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6431300 0.83 DBH (0.37) DBHMAOAALDH1A1ALOX15HSD17B10
SCHEMBL4652146 0.76
SCHEMBL11691899 0.74 DBH (0.33) DBHMAOAALDH1A1ALOX15HSD17B10
SCHEMBL11218287 0.74 TSHR (0.38) ALDH1A1TDP1LMNATSHRCA9
SCHEMBL1515006 0.74 CA12 (0.31) CA9CA12PARP1
SCHEMBL6362215 0.74
SCHEMBL1534020 0.74 CYP1A2 (0.33) ALDH1A1TDP1CA2CA1TSHR
SCHEMBL4420230 0.74 CES2 (0.33) CA9CA12PARP1
SCHEMBL3293588 0.74 ALDH1A1 (0.43) ALDH1A1ALOX15HSD17B10TDP1HPGD
SCHEMBL1153261 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014025993-A1 INHIBITORS OF D-AMINO ACID OXIDASE THE JOHNS HOPKINS UNIVERSITY (US) 2014-02-13 WO disclosed
US-6355805-B1 MULTIBINDING COMPOUNDS USEFUL IN TREATMENT AND PREVENTION OF METABOLIC DISORDERS SUCH AS OBESITY AND DIABETES ADVANCED MEDICINE, INC. 2002-03-12 US disclosed
EP-1085894-A1 BETA 3-ADRENERGIC RECEPTOR AGONISTS Advanced Medicine, Inc. (US) 2001-03-28 EP disclosed
WO-1999064053-A1 β3-ADRENERGIC RECEPTOR AGONISTS ADVANCED MEDICINE, INC. (US) 1999-12-16 WO disclosed
EP-0003758-A1 Etherified hydroxy-benzodiheterocycles and their acid addition salts, process for their preparation and pharmaceutical compositions containing them CIBA-GEIGY AG (CH) 1979-09-05 EP disclosed