SCHEMBL1534020

SCHEMBL1534020

Cc1cccc2c1=NC(=O)N=2

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.33
CYP2A6 P11509 1/20 0.33
ALDH1A1 P00352 2/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32
TSHR P16473 1/20 0.32
ACHE P22303 1/20 0.32
PARP1 P09874 4/20 0.32
ELANE P08246 3/20 0.32
TDP1 Q9NUW8 1/20 0.31
RPS6KA3 P51812 1/20 0.31
HCAR1 Q9BXC0 1/20 0.31
USP8 P40818 1/20 0.31
DAO P14920 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31748052 0.83 RPS6KA3 (0.37) CYP1A2CYP2A6ALDH1A1CA1CA2
SCHEMBL17427808 0.76 TDP2 (0.33) CYP1A2
SCHEMBL30417607 0.74 CYP1A2 (0.33) CYP1A2CYP2A6ALDH1A1CA1CA2
SCHEMBL3227957 0.74 TDP2 (0.35)
SCHEMBL7724583 0.74 DBH (0.37) CYP1A2ALDH1A1CA1CA2CA7
SCHEMBL25418829 0.74 CYP3A4 (0.33) ALDH1A1TSHRPARP1ELANETDP1
SCHEMBL1515006 0.74 CA12 (0.31) CA9PARP1
SCHEMBL11218287 0.74 TSHR (0.38) CYP1A2CYP2A6ALDH1A1CA9TSHR
SCHEMBL640435 0.74 CYP3A4 (0.33) ALDH1A1TSHRPARP1ELANETDP1
SCHEMBL11135354 0.74 CA1 (0.39) CYP2A6ALDH1A1CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 57 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104513494-A Preparation method for pigment orange 64 with high color intensity SHANGYU SHUNLIAN CHEMICAL CO LTD 2015-04-15 CN claimed
US-4122158-A FOR TREATMENT OF BURNS; BIODEGRADABLE HYDROPHOBIC POLYMER; SUSTAINED RELEASE ALZA CORPORATION (US) 1978-10-24 US claimed
US-20250388587-A1 TROPOMYOSIN RECEPTOR KINASE (TRK) DEGRADATION COMPOUNDS AND METHODS OF USE CULLGEN SHANGHAI INC (CN) 2025-12-25 US disclosed
US-20250059221-A1 STAT DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS, INC. 2025-02-20 US disclosed
US-20240417388-A1 BENZIMIDAZOLONE DERIVED INHIBITORS OF BCL6 CANCER RESEARCH TECH LTD (GB) 2024-12-19 US disclosed
US-20240400570-A1 TROPOMYOSIN RECEPTOR KINASE (TRK) DEGRADATION COMPOUNDS AND METHODS OF USE CULLGEN (SHANGHAI), INC. (CN) 2024-12-05 US disclosed
US-12077555-B2 STAT degraders and uses thereof KYMERA THERAPEUTICS, INC. (US) 2024-09-03 US disclosed
US-12065442-B2 Tropomyosin receptor kinase (TRK) degradation compounds and methods of use CULLGEN (SHANGHAI), INC. (CN) 2024-08-20 US disclosed
US-11969472-B2 Tropomyosin receptor kinase (TRK) degradation compounds and methods of use CULLGEN (SHANGHAI), INC. (CN) 2024-04-30 US disclosed
EP-4334307-A1 CDK2 DEGRADERS AND USES THEREOF Kymera Therapeutics, Inc. (US) 2024-03-13 EP disclosed
US-11746120-B2 Stat degraders and uses thereof KYMERA THERAPEUTICS, INC. (US) 2023-09-05 US disclosed
US-4287069-A BY MIXING SLUDGE WITH RESIDUES FORMED BY REACTING TOLUENE DIISOCYANATE WITH OTHER REACTIVE COMPOUNDS BAYER AKTIENGESELLSCHAFT (DE) 1981-09-01 US disclosed
EP-0027943-A1 Working-up process for cross-linked isocyanate-distillation residues containing urea groups, and the use of the products thus obtained as starting material in the production of plastics BAYER AG (DE) 1981-05-06 EP disclosed
US-4251638-A CONTAINING A REACTIVE FILLER WHICH IS DISTILLATION RESIDUE OF PRODUCTION OF TOLUENE DIISOCYANATE ISOMERS BAYER AKTIENGESELLSCHAFT (DE) 1981-02-17 US disclosed
US-4251401-A FOR PRODUCTION OF POLYURETHANES BAYER AKTIENGESELLSCHAFT (DE) 1981-02-17 US disclosed
EP-0011702-A1 TDI destillation residues dispersed in polyols and their use in a process for preparing polyurethane plastics BAYER AG (DE) 1980-06-11 EP disclosed
EP-0010675-A2 Working-up process of toluylen diisocyanate-distillation residues and use of the products thus obtained as mouldable material or as active fillers, in particular in the production of panels and shaped articles BAYER AG (DE) 1980-05-14 EP disclosed
EP-0010687-A1 Process for the production of polyurethanes from tuluylendiisocyanate residues and their use for preparing panels and moulded articles BAYER AG (DE) 1980-05-14 EP disclosed
US-4024125-A Dis-azo pigments deriving from bis-diazotized diamino-2-phenyl-benzazolones HOECHST AKTIENGESELLSCHAFT (DT) 1977-05-17 US disclosed
US-3987075-A ALKYL BENZENE SOLVENT OLIN CORPORATION (US) 1976-10-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11969472-B2 Tropomyosin receptor kinase (TRK) degradation compounds and methods of use MUSK, ERBB2, NTRK1 CYP1A2 4437/4885CYP2A6 4083/4885ALDH1A1 4113/4885
US-12077555-B2 STAT degraders and uses thereof STAT4, STAT1, STAT3 CYP1A2 486/4885CYP2A6 506/4885ALDH1A1 2465/4885
US-20250388587-A1 TROPOMYOSIN RECEPTOR KINASE (TRK) DEGRADATION COMPOUNDS AND METHODS OF USE ERBB2, MUSK, ERBB3 CYP1A2 4346/4885CYP2A6 2336/4885ALDH1A1 4483/4885
US-20250059221-A1 STAT DEGRADERS AND USES THEREOF STAT4, STAT1, STAT3 CYP1A2 486/4885CYP2A6 506/4885ALDH1A1 2465/4885
US-20240400570-A1 TROPOMYOSIN RECEPTOR KINASE (TRK) DEGRADATION COMPOUNDS AND METHODS OF USE MUSK, ERBB2, NTRK1 CYP1A2 4437/4885CYP2A6 4083/4885ALDH1A1 4113/4885
US-11746120-B2 Stat degraders and uses thereof STAT4, STAT1, STAT3 CYP1A2 486/4885CYP2A6 506/4885ALDH1A1 2465/4885
US-20240417388-A1 BENZIMIDAZOLONE DERIVED INHIBITORS OF BCL6 BCL6, BCL6B, BCL3 CYP1A2 2414/4885CYP2A6 1150/4885ALDH1A1 1654/4885
US-12065442-B2 Tropomyosin receptor kinase (TRK) degradation compounds and methods of use MUSK, NTRK1, ERBB2 CYP1A2 4053/4885CYP2A6 3652/4885ALDH1A1 3928/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.