SCHEMBL7724901

SCHEMBL7724901

CCc1cc(OC)c(C=O)cc1F

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.57
KDM4E B2RXH2 2/20 0.57
TSHR P16473 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
HPGD P15428 2/20 0.50
LMNA P02545 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
TAAR1 Q96RJ0 2/20 0.46
PRKDC P78527 2/20 0.43
MAPT P10636 2/20 0.42
ERN1 O75460 5/20 0.41
GAA P10253 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MEN1 O00255 1/20 0.39
POLB P06746 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP3A4 P08684 1/20 0.39
ALOX15 P16050 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20135982 0.86 ALDH1A1 (0.63) ALDH1A1KDM4ETSHRTDP1HPGD
SCHEMBL2432873 0.85 ALDH1A1 (0.47) ALDH1A1KDM4ETSHRTDP1HPGD
SCHEMBL668963 0.85 ALDH1A1 (0.67) ALDH1A1KDM4ETSHRTDP1HPGD
SCHEMBL26107991 0.83 ALDH1A1 (0.50) ALDH1A1KDM4ETSHRTDP1HPGD
SCHEMBL13618030 0.82 TAAR1 (0.53) TAAR1CYP3A4
SCHEMBL4813783 0.82 ALDH1A1 (0.68) ALDH1A1KDM4ETSHRTDP1HPGD
SCHEMBL29950688 0.82 ALDH1A1 (0.68) ALDH1A1KDM4ETSHRTDP1HPGD
SCHEMBL4071797 0.81 ALDH1A1 (0.67) ALDH1A1KDM4ETSHRTDP1HPGD
SCHEMBL7720458 0.80 TAAR1 (0.62) TAAR1CYP3A4
SCHEMBL20022271 0.80 ALDH1A1 (0.50) ALDH1A1KDM4ETSHRTDP1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1255396-C Carboxylic acid derivatives containing fused rings EISAI CO LTD (JP) 2006-05-10 CN disclosed
CN-1211361-C Carboxylic acid derivatives containing fused rings EISAI CO LTD (JP) 2005-07-20 CN disclosed
CN-1548428-A Carboxylic acid derivatives containing fused rings ������������ʽ���� 2004-11-24 CN disclosed
US-6358995-B1 AGONIST FOR RETINOIC ACID RECEPTORS; CAN BE SUBSTITUTED FOR RETINOIC ACID AS PREVENTIVE AND THERAPEUTIC DRUGS FOR VARIOUS DISEASES OR CANCERS, SUCH AS ACUTE PROMYELOCYTIC LEUKEMIA. EISAI CO., LTD. (JP) 2002-03-19 US disclosed
US-6121309-A SUCH AS 4-(2-(5-(7-FLUORO-4-TRIFLUOROMETHYLBENZOFURAN-2-YL)PYRROLYL)) BENZOIC ACID; RETINOIC ACID RECEPTOR AGONISM EISAI CO., LTD. (JP) 2000-09-19 US disclosed
US-6110959-A A RETINOIC ACID RECEPTOR AGONIST EISAI CO., LTD. (JP) 2000-08-29 US disclosed
CN-1214042-A Carboxylic acid derivatives containing fused rings EISAI CO LTD (JP) 1999-04-14 CN disclosed
EP-0889032-A1 FUSED-RING CARBOXYLIC ACID DERIVATIVES Eisai Co., Ltd. (JP) 1999-01-07 EP disclosed