SCHEMBL7724994

SCHEMBL7724994

COc1ccc2ccc(C#N)cc2c1C=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
AR P10275 3/20 0.42
ACHE P22303 1/20 0.40
CYP1A2 P05177 1/20 0.40
MAPT P10636 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39
NCEH1 Q6PIU2 2/20 0.39
HPGDS O60760 1/20 0.38
ALPL P05186 2/20 0.38
IMPDH2 P12268 1/20 0.38
IMPDH1 P20839 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TSHR P16473 1/20 0.38
GAA P10253 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19313483 0.81 IMPDH2 (0.47) ARIMPDH2IMPDH1ALDH1A1
SCHEMBL7336337 0.79 CYP1A2 (0.47) CA1CA2ARACHECYP1A2
SCHEMBL7336333 0.79 CYP1A2 (0.47) CA1CA2ARACHECYP1A2
Iodide SCHEMBL28325824 0.78 IMPDH2 (0.45) ARIMPDH2IMPDH1ALDH1A1
SCHEMBL19530936 0.78 ACHE (0.47) ACHECYP1A2MAPTCYP2C9CYP2C19
SCHEMBL7337530 0.78 AR (0.46) CA1CA2ARACHEMAPT
SCHEMBL5227187 0.78 MTNR1A (0.59) CA1CA2CYP1A2MAPTCYP2C9
SCHEMBL7723749 0.78 AR (0.50) CA1CA2ARACHENCEH1
Potassium Iodide SCHEMBL28325822 0.77 IMPDH2 (0.44) ARIMPDH2IMPDH1ALDH1A1
SCHEMBL7344856 0.76 AR (0.45) CA1CA2ARACHENCEH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6358995-B1 AGONIST FOR RETINOIC ACID RECEPTORS; CAN BE SUBSTITUTED FOR RETINOIC ACID AS PREVENTIVE AND THERAPEUTIC DRUGS FOR VARIOUS DISEASES OR CANCERS, SUCH AS ACUTE PROMYELOCYTIC LEUKEMIA. EISAI CO., LTD. (JP) 2002-03-19 US disclosed
US-6121309-A SUCH AS 4-(2-(5-(7-FLUORO-4-TRIFLUOROMETHYLBENZOFURAN-2-YL)PYRROLYL)) BENZOIC ACID; RETINOIC ACID RECEPTOR AGONISM EISAI CO., LTD. (JP) 2000-09-19 US disclosed
US-6110959-A A RETINOIC ACID RECEPTOR AGONIST EISAI CO., LTD. (JP) 2000-08-29 US disclosed
EP-0889032-A1 FUSED-RING CARBOXYLIC ACID DERIVATIVES Eisai Co., Ltd. (JP) 1999-01-07 EP disclosed