SCHEMBL7726523

SCHEMBL7726523

CC(C)(C)OC(=O)N1C[C@H](N(C(=O)CN)C(=O)OC(C)(C)C)C[C@H]1C(=O)Nc1ccc(Cc2ccccc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 5/20 0.41
POLB P06746 2/20 0.40
NPC1 O15118 1/20 0.40
PTPN1 P18031 1/20 0.40
HTRA1 Q92743 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
USP30 Q70CQ3 1/20 0.38
JAK2 O60674 1/20 0.38
JAK1 P23458 1/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
MCL1 Q07820 1/20 0.37
ABL1 P00519 2/20 0.37
BCR P11274 2/20 0.37
HSD11B1 P28845 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7722105 0.92 PTPN1 (0.40) HDAC8POLBNPC1PTPN1HTRA1
SCHEMBL7731725 0.91 HDAC8 (0.44) HDAC8POLBNPC1PTPN1HTRA1
SCHEMBL7727252 0.90 KDM4E (0.46) HDAC8POLBNPC1KDM4ELMNA
SCHEMBL7731479 0.90 HDAC8 (0.44) HDAC8POLBNPC1HTRA1CYP1A2
SCHEMBL7728192 0.88 POLB (0.47) HDAC8POLBNPC1PTPN1CYP1A2
SCHEMBL7725709 0.88 NPC1 (0.43) HDAC8POLBNPC1PTPN1HTRA1
SCHEMBL7728833 0.85 SIRT2 (0.47) HDAC8POLB
SCHEMBL7727754 0.84 POLB (0.44) HDAC8POLBNPC1CYP1A2CYP3A4
SCHEMBL7729236 0.81 HDAC4 (0.41) HDAC8POLBNPC1CYP1A2CYP3A4
SCHEMBL7728738 0.81 KDM4E (0.46) POLBJAK2MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6399629-B1 PYRROLIDINES AND PIPERIDINES FOR TREATING MICROBIAL INFECTIONS BY REDUCING EXPORT OF COADMINISTERED ANTIMICROBIAL AGENT OR COMPOUND SYNTHESIZED BY MICROBES FOR THEIR GROWTH; REDUCING IN VIVO AVAILABILITY MICROCIDE PHARMACEUTICALS, INC. 2002-06-04 US disclosed