SCHEMBL7728351

SCHEMBL7728351

CC(C)(C)c1ccc2oc(C(O)[C@@H](CCc3ccccc3)NC(=O)[C@H]3C[C@H](CN)CN3)nc2c1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSS P25774 3/20 0.44
CTSL P07711 2/20 0.44
CTSB P07858 2/20 0.44
CTSK P43235 2/20 0.44
F2 P00734 9/20 0.38
MASP2 O00187 4/20 0.37
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
CTSC P53634 1/20 0.33
CTSD P07339 1/20 0.32
BACE1 P56817 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7723243 0.78 CTSL (0.43) CTSSCTSLCTSBCTSKNPC1
SCHEMBL7732434 0.77 CTSL (0.43) CTSSCTSLCTSBCTSKNPC1
SCHEMBL7728635 0.77 F2 (0.35) CTSSCTSLCTSBCTSKF2
SCHEMBL21436251 0.77 F2 (0.35) CTSSCTSLCTSBCTSKF2
Trifluoroacetic Acid SCHEMBL7732038 0.75 CTSL (0.41) CTSSCTSLCTSBCTSKNPC1
SCHEMBL21436289 0.74 F2 (0.37) CTSSCTSLCTSBCTSKF2
SCHEMBL21436586 0.74 F2 (0.37) CTSSCTSLCTSBCTSKF2
SCHEMBL8142222 0.74 F2 (0.37) CTSSCTSLCTSBCTSKF2
SCHEMBL21436588 0.74 F2 (0.37) CTSSCTSLCTSBCTSKF2
SCHEMBL7728949 0.74 F2 (0.37) CTSSCTSLCTSBCTSKF2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6399629-B1 PYRROLIDINES AND PIPERIDINES FOR TREATING MICROBIAL INFECTIONS BY REDUCING EXPORT OF COADMINISTERED ANTIMICROBIAL AGENT OR COMPOUND SYNTHESIZED BY MICROBES FOR THEIR GROWTH; REDUCING IN VIVO AVAILABILITY MICROCIDE PHARMACEUTICALS, INC. 2002-06-04 US disclosed