SCHEMBL7729324

SCHEMBL7729324

COC(=O)[C@H]1C[C@H](N(C(=O)OC(C)(C)C)C(=O)[C@@H](O)CN)CN1C(=O)OC(C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.34
MMP2 P08253 1/20 0.34
ANPEP P15144 1/20 0.34
PEPD P12955 3/20 0.34
HTRA1 Q92743 1/20 0.34
XPNPEP1 Q9NQW7 1/20 0.33
NR1H2 P55055 2/20 0.33
NR1H3 Q13133 1/20 0.33
CYP1A2 P05177 1/20 0.33
POLB P06746 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
P2RX3 P56373 2/20 0.32
CETP P11597 1/20 0.31
CCR2 P41597 1/20 0.31
HSD11B1 P28845 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
PDE4B Q07343 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7727566 0.90 HTRA1 (0.34) HTRA1NR1H2CYP1A2POLBCYP3A4
SCHEMBL7733526 0.85 PTPN1 (0.39) PTPN1MMP2ANPEPPEPDHTRA1
SCHEMBL7726393 0.85 PTPN1 (0.39) PTPN1MMP2ANPEPPEPDHTRA1
SCHEMBL7733813 0.85 PTPN1 (0.39) PTPN1MMP2ANPEPPEPDHTRA1
SCHEMBL21285787 0.81 HSD11B1 (0.42) PTPN1MMP2ANPEPHTRA1NR1H2
SCHEMBL34474260 0.76 MMP2 (0.40) PTPN1MMP2ANPEPHTRA1NR1H2
SCHEMBL34474739 0.76 MMP2 (0.40) PTPN1MMP2ANPEPHTRA1NR1H2
SCHEMBL14915786 0.76 MMP2 (0.40) PTPN1MMP2ANPEPHTRA1NR1H2
SCHEMBL34474691 0.76 MMP2 (0.40) PTPN1MMP2ANPEPHTRA1NR1H2
SCHEMBL7727961 0.75 HSD17B10 (0.34) PTPN1HTRA1NR1H2CYP1A2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6399629-B1 PYRROLIDINES AND PIPERIDINES FOR TREATING MICROBIAL INFECTIONS BY REDUCING EXPORT OF COADMINISTERED ANTIMICROBIAL AGENT OR COMPOUND SYNTHESIZED BY MICROBES FOR THEIR GROWTH; REDUCING IN VIVO AVAILABILITY MICROCIDE PHARMACEUTICALS, INC. 2002-06-04 US disclosed