SCHEMBL7730052

SCHEMBL7730052

COc1ccc(N=CCC(C)C)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S100B P04271 1/20 0.45
ALDH1A1 P00352 2/20 0.42
ACHE P22303 1/20 0.42
CA12 O43570 2/20 0.41
CA2 P00918 2/20 0.41
CA9 Q16790 2/20 0.41
CA1 P00915 1/20 0.41
CA7 P43166 1/20 0.41
CA14 Q9ULX7 1/20 0.41
NOS3 P29474 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40
HTR3A P46098 1/20 0.40
HTR3D Q70Z44 1/20 0.40
HTR3C Q8WXA8 1/20 0.40
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
PKM P14618 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL709437 0.86 CYP2C9 (0.36) S100BALDH1A1SMN1; SMN2MAPTPTGS2
SCHEMBL7763844 0.79 S100B (0.49) S100BALDH1A1ACHECA12CA2
SCHEMBL12534124 0.79 S100B (0.49) S100BALDH1A1ACHECA12CA2
SCHEMBL11294036 0.76 ASF1A (0.40) ALDH1A1NOS3SMN1; SMN2NPC1MAPT
SCHEMBL22340706 0.76 S100B (0.38) S100BALDH1A1NOS3SMN1; SMN2HTR3E
SCHEMBL6560170 0.76 S100B (0.46) S100BALDH1A1ACHECA12CA2
SCHEMBL21565112 0.75 S100B (0.49) S100BALDH1A1ACHECA12CA2
SCHEMBL12616347 0.73 CA12 (0.55) S100BALDH1A1ACHECA12CA2
SCHEMBL9640860 0.73 CA12 (0.55) S100BALDH1A1ACHECA12CA2
SCHEMBL12617752 0.73 CA12 (0.55) S100BALDH1A1ACHECA12CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0690856-B1 ANTI-TUMOR COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, METHODS FOR PREPARATION THEREOF AND FOR TREATMENT UNIV NEW YORK STATE RES FOUND (US) 2002-12-04 EP disclosed
US-5705508-A FORMING TAXOL DERIVATIVES THE RESEARCH FOUNDATION OF STATE UNIVERSITY OF NEW YORK (US) 1998-01-06 US disclosed
US-5599820-A Anti-tumor compounds, pharmaceutical compositions, methods for preparation thereof and for treatment THE RESEARCH FOUNDATION OF STATE UNIVERSITY OF NEW YORK (US) 1997-02-04 US disclosed
US-5475011-A Anti-tumor compounds, pharmaceutical compositions, methods for preparation thereof and for treatment THE RESEARCH FOUNDATION OF STATE UNIVERSITY OF NEW YORK (US) 1995-12-12 US disclosed
US-5294737-A Hydrolysis, cyclization, condensation THE RESEARCH FOUNDATION STATE UNIVERSITY OF NEW YORK (US) 1994-03-15 US disclosed