SCHEMBL7733849

SCHEMBL7733849

COc1c(Cl)cc(F)cc1Br

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.43
CA4 P22748 2/20 0.43
HTR2A P28223 3/20 0.38
PTGS2 P35354 2/20 0.36
HSD17B10 Q99714 1/20 0.35
TPMT P51580 2/20 0.34
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
GAA P10253 1/20 0.34
POLB P06746 1/20 0.34
P2RX7 Q99572 1/20 0.34
TSHR P16473 1/20 0.33
APOBEC3A P31941 1/20 0.33
HTT P42858 1/20 0.33
APOBEC3G Q9HC16 1/20 0.33
CA1 P00915 1/20 0.33
CA6 P23280 1/20 0.33
NQO2 P16083 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1163205 0.84 CA2 (0.52) CA2CA4HTR2AHSD17B10TPMT
SCHEMBL3759267 0.84 ALDH1A1 (0.44) PTGS2HSD17B10TPMTALDH1A1KDM4E
SCHEMBL30407976 0.78 CA2 (0.46) CA2CA4HTR2AHSD17B10TPMT
SCHEMBL2415199 0.78 CA2 (0.46) CA2CA4HSD17B10TPMTALDH1A1
SCHEMBL4355782 0.78 CA2 (0.46) CA2CA4HTR2AHSD17B10TPMT
SCHEMBL31015937 0.78 PTGS2 (0.37) PTGS2TPMTALDH1A1KDM4EGAA
SCHEMBL1223114 0.78 PTGS2 (0.37) PTGS2TPMTALDH1A1KDM4EGAA
SCHEMBL12269187 0.77 CA2 (0.45) CA2CA4HTR2AHSD17B10TPMT
SCHEMBL10209878 0.77 TSHR (0.50) CA2CA4HTR2APTGS2POLB
SCHEMBL14217767 0.77 CA2 (0.45) CA2CA4HTR2AHSD17B10TPMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9580444-B2 Polycyclic pyrazolinone derivative and herbicide comprising same as effective component thereof SAGAMI CHEMICAL RESEARCH INSTITUTE (JP) 2017-02-28 US disclosed
US-9580444-B2 Polycyclic pyrazolinone derivative and herbicide comprising same as effective component thereof SAGAMI CHEMICAL RESEARCH INSTITUTE (JP) 2017-02-28 US disclosed
US-20160024110-A1 POLYCYCLIC PYRAZOLINONE DERIVATIVE AND HERBICIDE COMPRISING SAME AS EFFECTIVE COMPONENT THEREOF KAKEN PHARMACEUTICAL CO., LTD. (JP) 2016-01-28 US disclosed
US-20160024110-A1 POLYCYCLIC PYRAZOLINONE DERIVATIVE AND HERBICIDE COMPRISING SAME AS EFFECTIVE COMPONENT THEREOF KAKEN PHARMACEUTICAL CO., LTD. (JP) 2016-01-28 US disclosed
EP-2975040-A1 POLYCYCLIC PYRAZOLINONE DERIVATIVE AND HERBICIDE COMPRISING SAME AS EFFECTIVE COMPONENT THEREOF Sagami Chemical Research Institute (JP) 2016-01-20 EP disclosed
WO-2014142307-A1 POLYCYCLIC PYRAZOLINONE DERIVATIVE AND HERBICIDE COMPRISING SAME AS EFFECTIVE COMPONENT THEREOF 公益財団法人相模中央化学研究所 (JP) 2014-09-18 WO disclosed
CN-1127457-C Process for electrophilic aromatic substitution BROMINE COMPOUNDS LTD (IL) 2003-11-12 CN disclosed
US-6399835-B1 ALKYLATION, HALOGENATION USING AQUEOUS SOLUTION OF ZINC HALIDE BROMINE COMPOUNDS LTD. (IL) 2002-06-04 US disclosed
CN-1280555-A Process for electrophilic aromatic substitution BROMINE COMPOUNDS LTD (IL) 2001-01-17 CN disclosed
EP-1032549-A1 PROCESS FOR ELECTROPHILIC AROMATIC SUBSTITUTION Bromine Compounds Ltd. (IL) 2000-09-06 EP disclosed
WO-1999019275-A1 PROCESS FOR ELECTROPHILIC AROMATIC SUBSTITUTION BROMINE COMPOUNDS LTD. (IL) 1999-04-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160024110-A1 POLYCYCLIC PYRAZOLINONE DERIVATIVE AND HERBICIDE COMPRISING SAME AS EFFECTIVE COMPONENT THEREOF DDT, PDHX, CYP4X1 CA2 1003/4885CA4 969/4885HTR2A 2936/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.