SCHEMBL7734258

SCHEMBL7734258

Cc1cnn(-c2ccc(N)cc2CN(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)c1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 1/20 0.35
CYP46A1 Q9Y6A2 3/20 0.34
GRM2 Q14416 2/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CG P48736 1/20 0.34
HCRTR2 O43614 2/20 0.32
CPB2 Q96IY4 8/20 0.32
NR1H2 P55055 1/20 0.32
HCRTR1 O43613 1/20 0.32
NTRK1 P04629 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27559418 0.84 TDO2 (0.40) TDO2CYP46A1GRM2PIK3CAPIK3CG
SCHEMBL7740471 0.83 ITGA4 (0.36)
SCHEMBL7734182 0.83 GRM2 (0.33) CYP46A1GRM2PIK3CAPIK3CGNTRK1
SCHEMBL6682105 0.78 PRKCI (0.37) GRM2NR1H2
SCHEMBL12569696 0.77 PRKCI (0.38) GRM2NR1H2
SCHEMBL6681898 0.77 MAPT (0.47) NR1H2
SCHEMBL7246662 0.76 GAA (0.36) GRM2NR1H2
SCHEMBL6680044 0.76 HTT (0.48) NR1H2
SCHEMBL6674369 0.76 PRKCI (0.41) GRM2NR1H2
SCHEMBL24891920 0.75 GRM2 (0.36) GRM2NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6414005-B1 BRAIN DISORDERS; ALZHEIMER'S DISEASE; PARKINSON'S DISEASE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-07-02 US disclosed
EP-1043312-A1 HETEROCYCLIC COMPOUNDS HAVING NOS INHIBITORY ACTIVITIES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-10-11 EP disclosed