SCHEMBL7734182

SCHEMBL7734182

Cc1cnn(-c2ccc(NC(N)=S)cc2CN(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 2/20 0.33
NTRK1 P04629 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CG P48736 1/20 0.33
KDM4E B2RXH2 1/20 0.32
CYP1A2 P05177 3/20 0.32
GAA P10253 4/20 0.32
ALDH1A1 P00352 4/20 0.32
KMT2A Q03164 2/20 0.32
ALOX5AP P20292 1/20 0.32
MAPKAPK2 P49137 1/20 0.32
SYK P43405 1/20 0.32
AR P10275 1/20 0.31
CYP46A1 Q9Y6A2 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31
MEN1 O00255 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7734258 0.83 TDO2 (0.35) GRM2NTRK1PIK3CAPIK3CGCYP46A1
SCHEMBL6678474 0.81 ALDH1A1 (0.39) GRM2CYP1A2GAAALDH1A1KMT2A
SCHEMBL7739635 0.80 ALDH1A1 (0.37) GRM2CYP1A2GAAALDH1A1KMT2A
SCHEMBL6675178 0.80 KDM4E (0.44) KDM4EGAAALDH1A1KMT2AMAPT
SCHEMBL6682248 0.80 ALDH1A1 (0.40) GRM2CYP1A2GAAALDH1A1KMT2A
SCHEMBL6675695 0.79 ALDH1A1 (0.39) GRM2CYP1A2GAAALDH1A1KMT2A
SCHEMBL6675941 0.79 KDM4E (0.43) KDM4ECYP1A2GAAALDH1A1KMT2A
SCHEMBL7734178 0.79 NTRK1 (0.35) NTRK1PIK3CAPIK3CGKDM4ECYP1A2
SCHEMBL6681804 0.78 GRM2 (0.38) GRM2CYP1A2GAAALDH1A1KMT2A
SCHEMBL6678436 0.78 ALDH1A1 (0.40) GAAALDH1A1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6414005-B1 BRAIN DISORDERS; ALZHEIMER'S DISEASE; PARKINSON'S DISEASE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-07-02 US disclosed
EP-1043312-A1 HETEROCYCLIC COMPOUNDS HAVING NOS INHIBITORY ACTIVITIES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-10-11 EP disclosed