SCHEMBL7737053

SCHEMBL7737053

COc1cccc2c1OCCN2CCO

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.49
SLC6A4 P31645 1/20 0.49
KCNH2 Q12809 1/20 0.42
PTGIR P43119 1/20 0.42
NR3C1 P04150 1/20 0.39
PGR P06401 1/20 0.39
NR3C2 P08235 1/20 0.39
DRD2 P14416 2/20 0.38
DRD3 P35462 1/20 0.38
MAPT P10636 1/20 0.38
TSHR P16473 2/20 0.37
CYP2D6 P10635 1/20 0.37
CTNNB1 P35222 1/20 0.37
WNT3A P56704 1/20 0.37
ALPL P05186 1/20 0.37
ADRA1D P25100 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36
NOTUM Q6P988 1/20 0.36
AKR1C3 P42330 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5908138 0.83 PTGIR (0.50) HTR1ASLC6A4PTGIRTSHRALPL
SCHEMBL7736507 0.81 PTGIR (0.63) HTR1ASLC6A4PTGIRTSHR
SCHEMBL7729866 0.80 DRD2 (0.38) HTR1ASLC6A4PTGIRDRD2DRD3
SCHEMBL13545370 0.79 CYSLTR2 (0.40) HTR1ASLC6A4PTGIRMAPTTSHR
SCHEMBL8133224 0.74 KMT2A (0.56) HTR1ASLC6A4KCNH2MAPTTSHR
SCHEMBL18569479 0.74 DRD2 (0.41) HTR1ASLC6A4DRD2DRD3MAPT
SCHEMBL13383381 0.71 CYSLTR2 (0.43) HTR1ASLC6A4PTGIRTSHRNOTUM
SCHEMBL8572986 0.70 DRD2 (0.39) DRD2DRD3MAPTALPL
SCHEMBL6876623 0.69 DRD2 (0.42) DRD2DRD3MAPTNOTUM
SCHEMBL13681724 0.68 DRD2 (0.47) SLC6A4DRD2DRD3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407096-B1 1,4-BENZOTHIAZINE AND 1,4-BENZOXAZINE DERIVATIVES; HYPOTENSIVE, ANTIISCHEMIC, ANTIALLERGEN, ANTIASTHMATIC AND ANTICOAGULANT AGENTS; CARDIOVASCULAR DISORDERS TORAY INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1028113-A1 FUSED BENZENE HETEROCYCLE DERIVATIVES AND UTILIZATION THEREOF TORAY INDUSTRIES, INC. (JP) 2000-08-16 EP disclosed