SCHEMBL7737173

SCHEMBL7737173

Oc1ccc(F)c(F)c1I

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA3 P07451 1/20 0.39
CA6 P23280 1/20 0.39
CA5A P35218 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
CA5B Q9Y2D0 1/20 0.39
KDM4E B2RXH2 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
MPI P34949 1/20 0.38
CES2 O00748 2/20 0.36
CES1 P23141 2/20 0.36
IDO1 P14902 1/20 0.33
HSD17B1 P14061 2/20 0.31
HSD17B2 P37059 2/20 0.31
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
MEP1B Q16820 1/20 0.30
BCHE P06276 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16089554 0.79 CA3 (0.39) CA3CA6CA5ACA9CA14
SCHEMBL25346822 0.79 CA3 (0.39) CA3CA6CA5ACA9CA14
SCHEMBL13488 0.77 CES2 (0.36) CES2CES1
SCHEMBL12804172 0.75 DAO (0.38) CA3CA6CA5ACA9CA14
SCHEMBL24978467 0.75 TP53 (0.36) KDM4EESR1ESR2
SCHEMBL24252843 0.75 CYP3A4 (0.42) KDM4EHSD17B1HSD17B2ESR2
SCHEMBL30467752 0.75 CYP3A4 (0.42) KDM4EHSD17B1HSD17B2ESR2
SCHEMBL155976 0.75 CES2 (0.46) CA3CA6CA5ACA9CA14
SCHEMBL361051 0.73 PIM1 (0.41) CA3CA6CA5ACA9CA14
SCHEMBL5506954 0.72 ADRA2A (0.45) CA3CA6CA5ACA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3080132-A1 BROMODOMAIN INHIBITORS AbbVie Inc. (US) 2016-10-19 EP disclosed
CN-105980392-A Bromodomain inhibitors 艾伯维公司 2016-09-28 CN disclosed
WO-2015085925-A1 BROMODOMAIN INHIBITORS ABBVIE INC. (US) 2015-06-18 WO disclosed
US-6413448-B1 ESTERS; DOPANTS; LONGER CHIRAL SMECTIC PHASE PITCH; HIGHER TILT ANGLE; LOWER VISCOSITY; CRYSTALLIZATION SUPPRESSION; IMPROVED SOLUBILITY; BROADER C* PHASE TEMPERATURE RANGE DISPLAYTECH, INC. 2002-07-02 US disclosed
WO-2000065801-A9 CYCLOHEXYL- AND CYCLOHEXENYL-SUBSTITUTED LIQUID CRYSTALS WITH LOW BIREFRINGENCE DISPLAYTECH INC (US) 2001-04-12 WO disclosed
WO-2000065801-A1 CYCLOHEXYL- AND CYCLOHEXENYL-SUBSTITUTED LIQUID CRYSTALS WITH LOW BIREFRINGENCE DISPLAYTECH, INC. (US) 2000-11-02 WO disclosed