SCHEMBL7739145

SCHEMBL7739145

C=CCc1ccc(C(C)=C(NC(C)=O)C(=O)O)c([SiH](C)C)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.36
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
TDP1 Q9NUW8 2/20 0.34
CYP3A4 P08684 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
KDM4E B2RXH2 4/20 0.33
XDH P47989 1/20 0.33
LMNA P02545 1/20 0.33
ALOX5 P09917 3/20 0.33
MAPT P10636 2/20 0.33
PPARA Q07869 2/20 0.33
ALDH1A1 P00352 4/20 0.33
PPARG P37231 2/20 0.33
PPARD Q03181 2/20 0.33
ALDH2 P05091 1/20 0.33
GAA P10253 1/20 0.33
GABRA1 P14867 1/20 0.33
AKR1B1 P15121 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7737555 0.81 PTGS1 (0.35) PTGS1MEN1KMT2ATDP1CYP3A4
SCHEMBL7739194 0.79 XDH (0.42) PTGS1MEN1KMT2ATDP1CYP3A4
SCHEMBL7738425 0.79 PTGS1 (0.44) PTGS1MEN1KMT2ATDP1CYP3A4
SCHEMBL7737541 0.76 PTGS1 (0.45) PTGS1MEN1KMT2ATDP1CYP3A4
SCHEMBL7736596 0.73 MEN1 (0.33) MEN1KMT2AKDM4ELMNAMAPT
SCHEMBL7732390 0.69 PPARA (0.40) PTGS1MEN1KMT2ATDP1CYP3A4
SCHEMBL7738413 0.68 PPARA (0.36) PTGS1MEN1KMT2ATDP1CYP3A4
SCHEMBL7739200 0.66 PPARA (0.35) PTGS1MEN1KMT2ATDP1CYP3A4
SCHEMBL7737533 0.65 ALDH1A1 (0.41) PTGS1MEN1KMT2ATDP1CYP3A4
SCHEMBL7732384 0.65 XDH (0.44) PTGS1MEN1KMT2ACYP3A4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6416861-B1 COMBINATORIAL CHEMISTRY NORTHWESTERN UNIVERSITY 2002-07-09 US disclosed
WO-2000049022-A2 ORGANOSILICON COMPOUNDS AND USES THEREOF NORTHWESTERN UNIVERSITY (US) 2000-08-24 WO disclosed