SCHEMBL7740552

SCHEMBL7740552

CCCCOC(=O)N1CCC=C(CI)C1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.47
LMNA P02545 1/20 0.47
POLB P06746 1/20 0.47
HRH2 P25021 2/20 0.39
HRH1 P35367 2/20 0.39
BCHE P06276 1/20 0.36
ALDH1A1 P00352 5/20 0.35
HPGD P15428 2/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
TDP1 Q9NUW8 2/20 0.35
KDM4E B2RXH2 1/20 0.35
TSHR P16473 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ESR1 P03372 1/20 0.35
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
NPC1 O15118 1/20 0.34
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7745371 0.84 SMN1; SMN2 (0.45) SMN1; SMN2LMNAPOLBHRH2HRH1
SCHEMBL27563812 0.80 LMNA (0.48) SMN1; SMN2LMNAPOLBHRH2HRH1
SCHEMBL9627031 0.78 SMN1; SMN2 (0.50) SMN1; SMN2LMNAPOLBHRH2HRH1
SCHEMBL6659330 0.76 ESR2 (0.43) SMN1; SMN2LMNAALDH1A1KMT2AMEN1
SCHEMBL9457164 0.75 SMN1; SMN2 (0.44) SMN1; SMN2LMNAPOLBHRH2HRH1
SCHEMBL6661592 0.75 MEN1 (0.52) SMN1; SMN2HRH2HRH1ALDH1A1HPGD
SCHEMBL574934 0.75 SMN1; SMN2 (0.63) SMN1; SMN2LMNAPOLBHRH2HRH1
Iodide SCHEMBL7860350 0.74 MEN1 (0.51) SMN1; SMN2HRH2HRH1ALDH1A1HPGD
SCHEMBL30643716 0.74 HRH2 (0.47) SMN1; SMN2LMNAPOLBHRH2HRH1
SCHEMBL29736653 0.73 SMN1; SMN2 (0.44) SMN1; SMN2LMNAPOLBHRH2HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1080075-A4 PIPERIDIDINYL AND N-AMIDINOPIPERIDINYL DERIVATIVES AVENTIS PHARM PROD INC (US) 2001-06-27 EP disclosed
EP-1080075-A1 PIPERIDIDINYL AND N-AMIDINOPIPERIDINYL DERIVATIVES Aventis Pharmaceuticals Products Inc. (US) 2001-03-07 EP disclosed
WO-1999048870-A1 PIPERIDIDINYL AND N-AMIDINOPIPERIDINYL DERIVATIVES AVENTIS PHARMACEUTICALS PRODUCTS INC. (US) 1999-09-30 WO disclosed