SCHEMBL7742775

SCHEMBL7742775

CCC(C)OP(=O)(O)c1cc2cc(-c3ccc([N+](=O)[O-])cc3)c(Cl)cc2[nH]c1=O

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.40
GSK3B P49841 1/20 0.40
PGR P06401 1/20 0.34
GRIN1 Q05586 2/20 0.33
PRKAB2 O43741 1/20 0.33
PRKAG1 P54619 1/20 0.33
PRKAA2 P54646 1/20 0.33
PRKAA1 Q13131 1/20 0.33
PRKAG3 Q9UGI9 1/20 0.33
PRKAG2 Q9UGJ0 1/20 0.33
PRKAB1 Q9Y478 1/20 0.33
NPBWR1 P48145 1/20 0.33
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
GRIN2A Q12879 1/20 0.33
GRIN2B Q13224 1/20 0.33
GRIN2C Q14957 1/20 0.33
GRIN3A Q8TCU5 1/20 0.33
TYMS P04818 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7734973 0.91 GRIN2D (0.37) PGRGRIN1GRIN2DGRIN3BGRIN2A
SCHEMBL7741122 0.88 PRKAG1 (0.38) CYP1A2GSK3BGRIN1PRKAB2PRKAG1
SCHEMBL7739851 0.87 PRKAG1 (0.38) CYP1A2PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL7739647 0.87 PRKAG1 (0.38) CYP1A2GSK3BPRKAB2PRKAG1PRKAA2
SCHEMBL7740615 0.87 PRKAG1 (0.36) CYP1A2GSK3BPRKAB2PRKAG1PRKAA2
SCHEMBL7741420 0.86 CHRNA7 (0.36) CYP1A2PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL7740618 0.85 PTGES (0.38) GRIN1PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL7741121 0.85 IDH1 (0.36) PGRGRIN1PRKAB2PRKAG1PRKAA2
SCHEMBL6922994 0.84 CA12 (0.37) GRIN1GRIN2DGRIN3BGRIN2AGRIN2B
SCHEMBL7741259 0.84 PRKAG1 (0.35) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6420386-B1 SPINAL TRAUMATISM, EPILEPSY, CHRONIC NEURODEGENERATIVE DISEASES SUCH AS ALZHEIMER'S DISEASE, SCHIZOPHRENIA, LATERAL AMYOTROPHIC SCLEROSIS OR HUNTINGTON'S CHOREA. LES LABORATORIES SERVIER (FR) 2002-07-16 US disclosed