SCHEMBL7744000

SCHEMBL7744000

CC[C@@H](C)N1C(=O)C(NC(=O)Cc2ccc(C(F)(F)F)cc2C(F)(F)F)N=C(C2CC2)c2ccccc21

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.55
CCKBR P32239 11/20 0.37
XIAP P98170 1/20 0.37
PSEN1 P49768 2/20 0.36
PSEN2 P49810 2/20 0.36
APH1B Q8WW43 2/20 0.36
NCSTN Q92542 2/20 0.36
APH1A Q96BI3 2/20 0.36
PSENEN Q9NZ42 2/20 0.36
CCKAR P32238 4/20 0.36
POLQ O75417 2/20 0.36
P2RX7 Q99572 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7744124 1.00 KCNH2 (0.55) KCNH2CCKBRXIAPPSEN1PSEN2
SCHEMBL7744593 0.88 KCNH2 (0.72) KCNH2CCKBRPSEN1PSEN2APH1B
SCHEMBL7744135 0.88 KCNH2 (0.72) KCNH2CCKBRPSEN1PSEN2APH1B
SCHEMBL7743998 0.84 KCNH2 (0.61) KCNH2CCKBR
SCHEMBL7744698 0.84 KCNH2 (0.47) KCNH2XIAPPOLQP2RX7
SCHEMBL8620108 0.84 KCNH2 (0.77) KCNH2CCKBR
SCHEMBL8760273 0.80 KCNH2 (0.75) KCNH2CCKBRPSEN1PSEN2APH1B
SCHEMBL7743995 0.78 KCNH2 (0.36) KCNH2CCKBRXIAPPSEN1PSEN2
SCHEMBL7744120 0.78 KCNH2 (0.36) KCNH2CCKBRXIAPPSEN1PSEN2
SCHEMBL7965787 0.74 KCNH2 (0.85) KCNH2CCKBRCCKAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001010216-A1 ANTIARRHYTHMIC COMPOUNDS MERCK & CO., INC. (US) 2001-02-15 WO disclosed