SCHEMBL7743995

SCHEMBL7743995

CC[C@@H](C)N1C(=O)C(N(C(C)=O)c2ccc(C(F)(F)F)cc2C(F)(F)F)N=C(C2CC2)c2ccccc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.36
XIAP P98170 4/20 0.34
GALR3 O60755 1/20 0.33
CCKBR P32239 6/20 0.32
KLRK1 P26718 1/20 0.32
MICA Q29983 1/20 0.32
RAET1L Q5VY80 1/20 0.32
SCN9A Q15858 1/20 0.32
CCKAR P32238 2/20 0.31
BDKRB1 P46663 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
PDE2A O00408 1/20 0.31
PSEN1 P49768 2/20 0.31
PSEN2 P49810 2/20 0.31
APH1B Q8WW43 2/20 0.31
NCSTN Q92542 2/20 0.31
APH1A Q96BI3 2/20 0.31
PSENEN Q9NZ42 2/20 0.31
UBE2M P61081 1/20 0.30
DCUN1D1 Q96GG9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7744120 1.00 KCNH2 (0.36) KCNH2XIAPGALR3CCKBRKLRK1
SCHEMBL7744591 0.87 KCNH2 (0.45) KCNH2CCKBRCCKARPSEN1PSEN2
SCHEMBL7744132 0.87 KCNH2 (0.45) KCNH2CCKBRCCKARPSEN1PSEN2
SCHEMBL7744126 0.86 CCKBR (0.42) KCNH2CCKBRKLRK1MICARAET1L
SCHEMBL7744000 0.78 KCNH2 (0.55) KCNH2XIAPCCKBRCCKARPSEN1
SCHEMBL7744124 0.78 KCNH2 (0.55) KCNH2XIAPCCKBRCCKARPSEN1
SCHEMBL7744698 0.70 KCNH2 (0.47) KCNH2XIAPGALR3SCN9A
SCHEMBL7744588 0.68 CCKBR (0.44) KCNH2CCKBRBDKRB1
SCHEMBL7744135 0.67 KCNH2 (0.72) KCNH2CCKBRCCKARPSEN1PSEN2
SCHEMBL7744593 0.67 KCNH2 (0.72) KCNH2CCKBRCCKARPSEN1PSEN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001010216-A1 ANTIARRHYTHMIC COMPOUNDS MERCK & CO., INC. (US) 2001-02-15 WO disclosed