SCHEMBL7744698

SCHEMBL7744698

CC[C@H](C)N1C(=O)C(NC(=O)Cc2ccc(C(F)(F)F)cc2C(F)(F)F)C=C(C2CC2)c2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.47
XIAP P98170 3/20 0.37
POLQ O75417 4/20 0.37
P2RX7 Q99572 6/20 0.37
SCN9A Q15858 2/20 0.35
EPHX2 P34913 1/20 0.35
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
GALR3 O60755 1/20 0.33
FPR1 P21462 1/20 0.33
FPR2 P25090 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7744128 0.87 KCNH2 (0.52) KCNH2XIAPPOLQP2RX7SCN9A
SCHEMBL7744000 0.84 KCNH2 (0.55) KCNH2XIAPPOLQP2RX7
SCHEMBL7744124 0.84 KCNH2 (0.55) KCNH2XIAPPOLQP2RX7
SCHEMBL7744593 0.79 KCNH2 (0.72) KCNH2
SCHEMBL7744135 0.79 KCNH2 (0.72) KCNH2
SCHEMBL7036498 0.72 KCNH2 (0.47) KCNH2XIAPPOLQP2RX7SCN9A
SCHEMBL8760273 0.71 KCNH2 (0.75) KCNH2
SCHEMBL7854689 0.70 KCNH2 (0.47) KCNH2POLQP2RX7SCN9A
SCHEMBL7036494 0.70 KCNH2 (0.57) KCNH2XIAPPOLQSCN9A
SCHEMBL7743998 0.70 KCNH2 (0.61) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001010216-A1 ANTIARRHYTHMIC COMPOUNDS MERCK & CO., INC. (US) 2001-02-15 WO disclosed