SCHEMBL7744128

SCHEMBL7744128

CCCN1C(=O)C(NC(=O)Cc2ccc(C(F)(F)F)cc2C(F)(F)F)C=C(C2CC2)c2ccccc21

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.52
CCKBR P32239 3/20 0.43
POLQ O75417 3/20 0.38
XIAP P98170 2/20 0.37
P2RX7 Q99572 4/20 0.36
EPHX2 P34913 1/20 0.36
SCN9A Q15858 2/20 0.35
ALDH1A1 P00352 1/20 0.35
CRHR1 P34998 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7744698 0.87 KCNH2 (0.47) KCNH2POLQXIAPP2RX7EPHX2
SCHEMBL7036499 0.81 KCNH2 (0.49) KCNH2CCKBRPOLQXIAPP2RX7
SCHEMBL7743998 0.79 KCNH2 (0.61) KCNH2CCKBR
SCHEMBL7854692 0.79 KCNH2 (0.49) KCNH2CCKBRPOLQXIAPP2RX7
SCHEMBL7036496 0.76 KCNH2 (0.57) KCNH2CCKBRPOLQXIAPSCN9A
SCHEMBL7744138 0.74 KCNH2 (0.80) KCNH2CCKBR
SCHEMBL8620108 0.73 KCNH2 (0.77) KCNH2CCKBRSCN9A
SCHEMBL7744124 0.73 KCNH2 (0.55) KCNH2CCKBRPOLQXIAPP2RX7
SCHEMBL7744000 0.73 KCNH2 (0.55) KCNH2CCKBRPOLQXIAPP2RX7
SCHEMBL7965787 0.72 KCNH2 (0.85) KCNH2CCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001010216-A1 ANTIARRHYTHMIC COMPOUNDS MERCK & CO., INC. (US) 2001-02-15 WO disclosed