SCHEMBL7744317

SCHEMBL7744317

CC(=O)OC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@@]2(O)C(C)(C)[C@@]12O

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.52
ADORA3 P0DMS8 1/20 0.51
HSP90B1 P14625 1/20 0.46
PI4KA P42356 1/20 0.46
PI4K2B Q8TCG2 1/20 0.46
PI4K2A Q9BTU6 1/20 0.46
PI4KB Q9UBF8 1/20 0.46
RXFP1 Q9HBX9 1/20 0.44
AHCY P23526 7/20 0.44
P2RX1 P51575 1/20 0.43
P2RX3 P56373 1/20 0.43
P2RX4 Q99571 1/20 0.43
GSK3A P49840 2/20 0.43
RPS6KA3 P51812 2/20 0.43
MAPK14 Q16539 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25408738 1.00 ADORA2A (0.52) ADORA2AADORA3HSP90B1PI4KAPI4K2B
SCHEMBL6222357 0.85 ADORA2A (0.50) ADORA2AADORA3HSP90B1PI4KAPI4K2B
SCHEMBL2821282 0.85 ADORA2A (0.58) ADORA2AADORA3HSP90B1PI4KAPI4K2B
SCHEMBL19692161 0.84 ADORA2A (0.58) ADORA2AADORA3PI4KAPI4K2BPI4K2A
SCHEMBL1078828 0.84 ADORA2A (0.64) ADORA2AADORA3PI4KAPI4K2BPI4K2A
SCHEMBL11040343 0.84 ADORA2A (0.58) ADORA2AADORA3PI4KAPI4K2BPI4K2A
SCHEMBL28156591 0.84 ADORA2A (0.64) ADORA2AADORA3PI4KAPI4K2BPI4K2A
SCHEMBL8943715 0.83 ADORA2A (0.57) ADORA2AADORA3PI4KAPI4K2BPI4K2A
SCHEMBL5554234 0.83 ADORA2A (0.56) ADORA2AADORA3PI4KAPI4K2BPI4K2A
SCHEMBL9054202 0.82 ADORA2A (0.55) ADORA2AADORA3HSP90B1PI4KAPI4K2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0708781-B1 A 3 ADENOSINE RECEPTOR AGONISTS USA (US) 2001-10-04 EP disclosed
US-5773423-A XANTHINE RIBOSIDES THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1998-06-30 US disclosed
EP-0708781-A1 A 3 ADENOSINE RECEPTOR AGONISTS THE UNITED STATES OF AMERICA, as represented by THE SECRETARY, Department of Health and Human Services (US) 1996-05-01 EP disclosed
WO-1995002604-A1 A3 ADENOSINE RECEPTOR AGONISTS THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1995-01-26 WO disclosed