SCHEMBL7744409

SCHEMBL7744409

CCCCCc1n[nH]c2cccc(Cc3ccccc3)c12

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
NPC1 O15118 1/20 0.41
TLR8 Q9NR97 3/20 0.41
CYP2C9 P11712 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
HPGD P15428 2/20 0.40
ALOX12 P18054 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
POLB P06746 1/20 0.38
CETP P11597 1/20 0.38
TDP1 Q9NUW8 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CYP19A1 P11511 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3049376 0.86 LIPG (0.39) CETPTDP1L3MBTL1
SCHEMBL7746874 0.82 CYP2C9 (0.39) ALDH1A1NPC1CYP2C9CYP1A2CYP3A4
SCHEMBL27807083 0.76 PARP1 (0.39) CETPTDP1L3MBTL1
SCHEMBL6854925 0.73 GAA (0.51) CYP2C9CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL5315808 0.73 CYP1A2 (0.48) CYP2C9CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL5312171 0.72 CYP1A2 (0.44) ALDH1A1CYP2C9CYP1A2CYP3A4CYP2D6
SCHEMBL2876088 0.72 MEN1 (0.45) ALDH1A1NPC1CYP1A2CYP3A4CYP2C19
SCHEMBL22471642 0.71 HTR2A (0.57) TLR8
SCHEMBL29117330 0.71 MEN1 (0.47) ALDH1A1CYP1A2CYP3A4HPGDCETP
SCHEMBL3264340 0.71 TDP1 (0.38) ALDH1A1NPC1HPGDALOX12SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1252156-A1 BLOCKADE OF VOLTAGE DEPENDENT SODIUM CHANNELS University College London (GB) 2002-10-30 EP disclosed
WO-2001057024-A1 BLOCKADE OF VOLTAGE DEPENDENT SODIUM CHANNELS UNIVERSITY COLLEGE LONDON (GB) 2001-08-09 WO disclosed