SCHEMBL7744628

SCHEMBL7744628

Oc1ccc(C2=CCNCC2)cc1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
QDPR P09417 5/20 1.00
HTR2C P28335 8/20 0.58
SIGMAR1 Q99720 2/20 0.58
APP P05067 1/20 0.45
ESR1 P03372 1/20 0.42
ESR2 Q92731 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31367896 1.00 QDPR (1.00) QDPRHTR2CSIGMAR1APPESR1
SCHEMBL27866836 0.85 QDPR (0.73) QDPRHTR2CSIGMAR1
SCHEMBL17397697 0.85 QDPR (0.73) QDPRHTR2CSIGMAR1
SCHEMBL10827686 0.81 QDPR (0.69) QDPRAPP
SCHEMBL10407313 0.81 QDPR (1.00) QDPRHTR2CSIGMAR1
SCHEMBL8380936 0.81 QDPR (1.00) QDPRHTR2CSIGMAR1ESR1ESR2
Hydrochloric Acid SCHEMBL10353907 0.80 QDPR (0.67) QDPRHTR2CAPP
Hydrochloric Acid SCHEMBL17455197 0.79 QDPR (0.96) QDPRHTR2CSIGMAR1ESR1ESR2
SCHEMBL21228136 0.77 HTR2C (0.66) QDPRHTR2CSIGMAR1ESR1ESR2
SCHEMBL29914651 0.77 HTR2C (0.66) QDPRHTR2CSIGMAR1ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5502050-A DIHYDROXYPHENYL-SUBSTITITED PYRIDINES OR QUINONES, HYPERTENSIVE AGENTS CORNELL RESEARCH FOUNDATION, INC. (US) 1996-03-26 US claimed
EP-0730451-A4 BLOCKING UTILIZATION OF TETRAHYDROBIOPTERIN TO BLOCK INDUCTION OF NITRIC OXIDE SYNTHESIS CORNELL RES FOUNDATION INC (US) 2001-11-28 EP disclosed
US-5874433-A Blocking utilization of tetrahydrobiopterin to block induction of nitric oxide synthesis CORNELL RESEARCH FOUNDATION, INC. (US) 1999-02-23 US disclosed
US-5874433-A Blocking utilization of tetrahydrobiopterin to block induction of nitric oxide synthesis CORNELL RESEARCH FOUNDATION, INC. (US) 1999-02-23 US disclosed
EP-0730451-A1 BLOCKING UTILIZATION OF TETRAHYDROBIOPTERIN TO BLOCK INDUCTION OF NITRIC OXIDE SYNTHESIS CORNELL RESEARCH FOUNDATION, INC. (US) 1996-09-11 EP disclosed
US-5502050-A DIHYDROXYPHENYL-SUBSTITITED PYRIDINES OR QUINONES, HYPERTENSIVE AGENTS CORNELL RESEARCH FOUNDATION, INC. (US) 1996-03-26 US disclosed
US-5502050-A DIHYDROXYPHENYL-SUBSTITITED PYRIDINES OR QUINONES, HYPERTENSIVE AGENTS CORNELL RESEARCH FOUNDATION, INC. (US) 1996-03-26 US disclosed
WO-1995014468-A1 BLOCKING UTILIZATION OF TETRAHYDROBIOPTERIN TO BLOCK INDUCTION OF NITRIC OXIDE SYNTHESIS CORNELL RESEARCH FOUNDATION INC. (US) 1995-06-01 WO disclosed