SCHEMBL7745294

SCHEMBL7745294

COc1cc(-c2ccccc2C(N)=O)cc2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.49
SLC6A2 P23975 1/20 0.46
SLC6A4 P31645 1/20 0.46
SLC6A3 Q01959 1/20 0.46
KDM4E B2RXH2 3/20 0.45
ALDH1A1 P00352 3/20 0.45
GAA P10253 1/20 0.45
ERN1 O75460 2/20 0.45
PARP15 Q460N3 1/20 0.44
PARP10 Q53GL7 1/20 0.44
PARP1 P09874 4/20 0.43
DHODH Q02127 2/20 0.43
CDC7 O00311 1/20 0.42
CHEK1 O14757 1/20 0.42
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA2B P29275 1/20 0.41
ADORA1 P30542 1/20 0.41
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10316385 0.82 HTT (0.57) BCAT2ALDH1A1ERN1PARP1CDC7
SCHEMBL7762502 0.81 BCAT2 (0.56) BCAT2SLC6A2SLC6A4SLC6A3KDM4E
SCHEMBL5023244 0.78 PARP1 (0.50) SLC6A2SLC6A4SLC6A3KDM4EALDH1A1
SCHEMBL29456755 0.78 KIT (0.44) ALDH1A1ADORA2AMEN1POLBMAPT
SCHEMBL8197756 0.77 NQO1 (0.54) KDM4EALDH1A1ERN1MAPTSMN1; SMN2
SCHEMBL28187515 0.76 BCAT2 (0.58) BCAT2SLC6A2SLC6A4SLC6A3KDM4E
SCHEMBL31281188 0.76 TSHR (0.49) KDM4EALDH1A1PARP15PARP10PARP1
SCHEMBL535683 0.76 TSHR (0.49) KDM4EALDH1A1PARP15PARP10PARP1
SCHEMBL21824069 0.75 ENPP2 (0.47) ALDH1A1ERN1MEN1MAPTKMT2A
Hydrochloric Acid SCHEMBL22445134 0.75 TSHR (0.47) KDM4EALDH1A1PARP15PARP10PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1129075-A1 N-ARYL(THIO)ANTHRANILIC ACID AMIDE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS VEGF RECEPTOR TYROSINE KINASE INHIBITORS Novartis AG (CH) 2001-09-05 EP disclosed
WO-2000027820-A1 N-ARYL(THIO)ANTHRANILIC ACID AMIDE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS VEGF RECEPTOR TYROSINE KINASE INHIBITORS NOVARTIS AG (CH) 2000-05-18 WO disclosed