SCHEMBL7745544

SCHEMBL7745544

O=C1CN(Cc2ccccc2)C(=O)C[N]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
DDB1 Q16531 1/20 0.42
CRBN Q96SW2 1/20 0.42
KMT2A Q03164 5/20 0.41
MEN1 O00255 4/20 0.41
POLB P06746 2/20 0.41
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
THRB P10828 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
F2 P00734 1/20 0.41
PLG P00747 1/20 0.41
ELANE P08246 1/20 0.41
CTSG P08311 1/20 0.41
CMA1 P23946 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1488276 0.79 L3MBTL1 (0.56) EPHX2L3MBTL1HPGDTSHRDDB1
SCHEMBL4892237 0.75 EPHX2 (0.45) EPHX2L3MBTL1HPGDTSHRDDB1
SCHEMBL9686511 0.73 L3MBTL1 (0.50) EPHX2L3MBTL1HPGDTSHRDDB1
SCHEMBL9058751 0.73 L3MBTL1 (0.59) EPHX2L3MBTL1HPGDTSHRDDB1
SCHEMBL5541824 0.72 L3MBTL1 (0.54) L3MBTL1HPGDTSHRDDB1CRBN
SCHEMBL10417429 0.72 L3MBTL1 (0.48) EPHX2L3MBTL1HPGDTSHRDDB1
SCHEMBL6858115 0.72 KMT2A (0.44) EPHX2L3MBTL1HPGDTSHRDDB1
SCHEMBL76982 0.71 ELANE (0.53) HPGDTSHRKMT2AMEN1POLB
SCHEMBL7142639 0.71 MEN1 (0.47) EPHX2L3MBTL1HPGDTSHRDDB1
SCHEMBL16085590 0.70 KMT2A (0.49) EPHX2L3MBTL1HPGDTSHRDDB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0819005-A4 2-ACYLAMINOPROPANAMIDES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2001-03-21 EP disclosed
US-5773441-A PRODRUGS; ANIMAL HUSBANDRY ELI LILLY AND COMPANY (US) 1998-06-30 US disclosed
EP-0819005-A1 2-ACYLAMINOPROPANAMIDES AS TACHYKININ RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 1998-01-21 EP disclosed
EP-0761220-A1 2-Acylaminopropanamides as growth hormone secretagogues ELI LILLY AND COMPANY (US) 1997-03-12 EP disclosed
WO-1997006803-A1 2-ACYLAMINOPROPANAMIDES AS GROWTH HORMONE SECRETAGOGUES ELI LILLY AND COMPANY (US) 1997-02-27 WO disclosed
US-5565568-A USEFUL IN TREATMENT OR PREVENTION OF A PHYSIOLOGICAL DISORDER ASSOCIATED WITH AN EXCESS OF TACHYKININS ELI LILLY AND COMPANY (US) 1996-10-15 US disclosed
WO-1996031214-A1 2-ACYLAMINOPROPANAMIDES AS TACHYKININ RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 1996-10-10 WO disclosed