SCHEMBL7746397

SCHEMBL7746397

Cc1csc(CC(=O)c2ccc(C)nc2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
LMNA P02545 1/20 0.39
KDM4C Q9H3R0 1/20 0.39
KMT2A Q03164 3/20 0.36
MAPT P10636 2/20 0.35
KCNQ3 O43525 1/20 0.35
KCNQ2 O43526 1/20 0.35
PRKAB2 O43741 1/20 0.34
PRKAG1 P54619 1/20 0.34
PRKAA2 P54646 1/20 0.34
PRKAA1 Q13131 1/20 0.34
PRKAG3 Q9UGI9 1/20 0.34
PRKAG2 Q9UGJ0 1/20 0.34
PRKAB1 Q9Y478 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7832355 0.82 NPC1 (0.47) KDM4ENPC1RAB9ASMN1; SMN2LMNA
SCHEMBL7832652 0.78 GSK3B (0.44) HDAC1HDAC6KDM4ENPC1RAB9A
SCHEMBL4778027 0.78 RAB9A (0.43) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL6168851 0.77 RAB9A (0.47) KDM4ENPC1RAB9ASMN1; SMN2LMNA
SCHEMBL7839557 0.75 NPC1 (0.51) HDAC1HDAC6NPC1RAB9ASMN1; SMN2
SCHEMBL7568236 0.75 CES2 (0.43) NPC1RAB9ALMNAKDM4CKMT2A
SCHEMBL7622865 0.75 TDP1 (0.50) KDM4ENPC1RAB9ASMN1; SMN2LMNA
SCHEMBL7846518 0.75 CES2 (0.43) HDAC1NPC1RAB9AKDM4CKMT2A
SCHEMBL7833284 0.71 KMT2A (0.48) HDAC1HDAC6KDM4ENPC1RAB9A
SCHEMBL2632670 0.71 HDAC1 (0.56) HDAC1HDAC6KDM4ESMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001029003-A1 PROCESS FOR THE PREPARATION OF 1-(6-METHYLPYRIDIN-3-YL)-2-(4-METHYLTHIOPHENYL)-ETHANONE AND ITS USE IN THE SYNTHESIS OF DIARYLPYRIDINES ZAMBON GROUP S.P.A. (IT) 2001-04-26 WO disclosed