SCHEMBL7747642

SCHEMBL7747642

COc1ccc(C2(N3CCN(C(Cc4ccc(C#N)cc4)c4cnc[nH]4)C(=C=O)C3)CCCCC2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 2/20 0.37
GRIN2B Q13224 2/20 0.37
GRIN2A Q12879 1/20 0.37
CYP19A1 P11511 4/20 0.36
SLC6A9 P48067 1/20 0.33
USP2 O75604 3/20 0.32
TSHR P16473 3/20 0.32
CYP2C9 P11712 3/20 0.32
CYP1A2 P05177 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
FPR2 P25090 3/20 0.32
FPR1 P21462 2/20 0.32
CYP3A4 P08684 3/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
CYP2D6 P10635 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
VNN1 O95497 1/20 0.31
MAOA P21397 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7555138 0.75 CYP3A4 (0.44) CYP19A1USP2TSHRCYP2C9CYP1A2
SCHEMBL3518402 0.68 OPRD1 (0.38) USP2TSHRCYP2C9CYP1A2SMN1; SMN2
SCHEMBL7850296 0.65 HRH3 (0.40) CYP19A1
SCHEMBL3517536 0.65 PIN1 (0.41) CYP19A1
SCHEMBL7134263 0.64 HRH3 (0.46) CYP19A1USP2
SCHEMBL7743502 0.64 MAPT (0.43) CYP19A1KMT2AALDH1A1
SCHEMBL3845496 0.64 FNTA (0.53) CYP19A1CYP3A4ALDH1A1
SCHEMBL5552211 0.64 HRH3 (0.41) CYP19A1
Hydrochloric Acid SCHEMBL7484921 0.64 HRH3 (0.45) CYP19A1USP2
Hydrochloric Acid SCHEMBL7528885 0.63 FNTA (0.53) CYP19A1CYP3A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000059930-A1 A METHOD OF TREATING CANCER MERCK & CO., INC. (US) 2000-10-12 WO claimed
WO-2001022963-A1 METHOD OF PREVENTING OSTEOPOROSIS MERCK & CO., INC. (US) 2001-04-05 WO disclosed