SCHEMBL7749765

SCHEMBL7749765

CN(C)C=Cc1cccnc1[N+](=O)[O-]

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.38
ALDH1A1 P00352 5/20 0.36
KMT2A Q03164 3/20 0.36
MAPT P10636 3/20 0.36
MEN1 O00255 2/20 0.36
MAPK1 P28482 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HTT P42858 2/20 0.35
POLB P06746 1/20 0.35
ESR2 Q92731 1/20 0.35
PDE10A Q9Y233 1/20 0.35
NCOA1 Q15788 1/20 0.35
NCOA3 Q9Y6Q9 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
RAB9A P51151 2/20 0.35
S1PR4 O95977 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8568414 0.79 RAB9A (0.40) NPC1ALDH1A1KMT2AMAPTMEN1
SCHEMBL8568417 0.79 RAB9A (0.40) NPC1ALDH1A1KMT2AMAPTMEN1
SCHEMBL2641785 0.79 MAPT (0.50) NPC1ALDH1A1KMT2AMAPTMEN1
SCHEMBL2641790 0.79 MAPT (0.50) NPC1ALDH1A1KMT2AMAPTMEN1
SCHEMBL9000495 0.78 PDE10A (0.40) NPC1ALDH1A1KMT2AMAPTMEN1
SCHEMBL27034756 0.76 TRIM24 (0.50) NPC1ALDH1A1KMT2AMAPTMEN1
SCHEMBL8561733 0.76 TAAR1 (0.47) NPC1ALDH1A1KMT2AMAPTMEN1
SCHEMBL8567625 0.76 KMT2A (0.41) NPC1ALDH1A1KMT2AMAPTMEN1
SCHEMBL8567627 0.76 KMT2A (0.41) NPC1ALDH1A1KMT2AMAPTMEN1
SCHEMBL1997660 0.75 PDE10A (0.45) NPC1ALDH1A1KMT2AMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0984932-A4 PROCESS FOR THE SYNTHESIS OF RIBONUCLEOTIDE REDUCTASE INHIBITORS 3-AP AND 3-AMP VION PHARMACEUTICALS INC (US) 2001-04-04 EP disclosed
EP-0984932-A1 PROCESS FOR THE SYNTHESIS OF RIBONUCLEOTIDE REDUCTASE INHIBITORS 3-AP AND 3-AMP Vion Pharmaceuticals, Inc. (US) 2000-03-15 EP disclosed
WO-1998051670-A1 PROCESS FOR THE SYNTHESIS OF RIBONUCLEOTIDE REDUCTASE INHIBITORS 3-AP AND 3-AMP VION PHARMACEUTICALS, INC. (US) 1998-11-19 WO disclosed
US-4625033-A 3-METHYL-4-NITROPYRIDINE-1-OXIDE CONDENSED TO ENAMINE, CATALYTIC REDUCTION CYCLIZATION SANOFI (FR) 1986-11-25 US disclosed