SCHEMBL7749970

SCHEMBL7749970

CP(=O)(O)C1=CCN(C(=O)OCC(Cl)(Cl)Cl)CC1

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RGS12 O14924 1/20 0.34
CYP3A4 P08684 1/20 0.34
TSHR P16473 1/20 0.34
GABRR1 P24046 1/20 0.34
GABRR2 P28476 1/20 0.34
MAPK1 P28482 1/20 0.34
BLM P54132 1/20 0.34
GNAI1 P63096 1/20 0.34
PMP22 Q01453 1/20 0.34
GRM5 P41594 2/20 0.31
GRM1 Q13255 2/20 0.31
SLC6A15 Q9H2J7 1/20 0.31
PDK4 Q16654 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14243233 0.81 SLC6A15 (0.36) CYP3A4MAPK1GRM5SLC6A15PDK4
SCHEMBL6678980 0.73 GRM5 (0.30) GRM5
SCHEMBL17243560 0.71 SLC6A15 (0.36) GRM5GRM1SLC6A15PDK4ALDH1A1
SCHEMBL3662063 0.70 ALDH1A1 (0.36) TSHRALDH1A1
SCHEMBL6322610 0.69 PRMT5 (0.47) CYP3A4TSHRALDH1A1LMNA
SCHEMBL11230779 0.68 ALDH1A1 (0.32) ALDH1A1
SCHEMBL11237397 0.68 DPP7 (0.38) TSHRALDH1A1LMNA
SCHEMBL21551284 0.68 GRM5 (0.56) CYP3A4GRM5ALDH1A1
SCHEMBL11480960 0.67 HPGD (0.43) CYP3A4TSHRGRM5GRM1ALDH1A1
SCHEMBL31166149 0.67 HDAC6 (0.47) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1000071-A4 NEUROLOGICALLY-ACTIVE COMPOUNDS POLYCHIP PHARMACEUTICALS PTY (AU) 2001-02-28 EP disclosed
EP-1000071-A1 NEUROLOGICALLY-ACTIVE COMPOUNDS Polychip Pharmaceuticals Pty. Ltd. (AU) 2000-05-17 EP disclosed
WO-1998058939-A1 NEUROLOGICALLY-ACTIVE COMPOUNDS POLYCHIP PHARMACEUTICALS PTY. LTD. (AU) 1998-12-30 WO disclosed