SCHEMBL7752953

SCHEMBL7752953

O=C(Nc1ccc([N+](=O)[O-])cc1C(=O)c1ccccc1)C(=O)c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 1/20 0.56
AKR1C4 P17516 1/20 0.54
AKR1C3 P42330 1/20 0.54
AKR1C2 P52895 1/20 0.54
AKR1C1 Q04828 1/20 0.54
CES2 O00748 2/20 0.52
MAPT P10636 6/20 0.52
LMNA P02545 4/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
POLB P06746 1/20 0.52
HTT P42858 1/20 0.52
CES1 P23141 1/20 0.51
CTSV O60911 1/20 0.51
CTSL P07711 1/20 0.51
ALDH1A1 P00352 2/20 0.49
GAA P10253 2/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
MYC P01106 1/20 0.46
MAX P61244 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7752904 0.86 AKR1C4 (0.67) PIN1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL19268076 0.86 PIN1 (0.53) PIN1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL6811878 0.85 CYP19A1 (0.59) PIN1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL8578400 0.83 MAPT (0.73) PIN1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL27346954 0.83 MAPT (0.56) PIN1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL6545840 0.82 AKR1C4 (0.52) PIN1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL11883066 0.82 ALDH1A1 (0.63) PIN1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL31541287 0.82 MEN1 (0.52) PIN1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL11157919 0.82 MEN1 (0.52) PIN1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL8568341 0.82 AKR1C4 (0.52) PIN1AKR1C4AKR1C3AKR1C2AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1068176-A1 CYSTEINE AMIDES AS FARNESYL TRANSFERASE INHIBITORS Jomaa, Hassan (DE) 2001-01-17 EP disclosed
WO-2000027803-A1 CYSTEINE AMIDES AS FARNESYL TRANSFERASE INHIBITORS JOMAA, HASSAN (DE) 2000-05-18 WO disclosed