SCHEMBL7753453

SCHEMBL7753453

COc1ccc(Cc2ccnc(N)n2)cc1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.55
CYP2D6 P10635 1/20 0.55
ATM Q13315 1/20 0.55
ROCK1 Q13464 1/20 0.50
NPSR1 Q6W5P4 1/20 0.48
POLB P06746 1/20 0.48
PDE3B Q13370 1/20 0.47
PDE3A Q14432 1/20 0.47
PDE10A Q9Y233 1/20 0.47
LTA4H P09960 2/20 0.46
TLR8 Q9NR97 1/20 0.45
TLR7 Q9NYK1 1/20 0.45
LMNA P02545 4/20 0.45
HPGD P15428 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
MPO P05164 1/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28993487 0.98 ALDH1A1 (0.54) ALDH1A1CYP2D6ATMROCK1NPSR1
SCHEMBL27943923 0.82 PDE3B (0.48) ALDH1A1CYP2D6ATMPOLBPDE3B
SCHEMBL30366498 0.81 ALDH1A1 (0.65) ALDH1A1CYP2D6ATMNPSR1POLB
Ammonia Solution, Strong SCHEMBL26627788 0.81 PDE3B (0.47) ALDH1A1CYP2D6ATMPOLBPDE3B
SCHEMBL2749244 0.80 ROCK1 (0.42) ROCK1TLR8TLR7
SCHEMBL11377589 0.78 ALDH1A1 (0.49) ALDH1A1CYP2D6ATMROCK1NPSR1
SCHEMBL1494107 0.78 AURKA (0.48) ROCK1POLBMPO
SCHEMBL30742723 0.77 DHFR (0.58) ALDH1A1SMN1; SMN2
Methyl Alcohol SCHEMBL29176241 0.77 L3MBTL1 (0.45) ROCK1POLBTLR8TLR7
SCHEMBL28133306 0.76 NPC1 (0.56) ALDH1A1CYP2D6LTA4HLMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1066266-A1 CYCLIN DEPENDENT KINASE INHIBITORS CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2001-01-10 EP disclosed
WO-1999050251-A2 CYCLIN DEPENDENT KINASE INHIBITORS CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 1999-10-07 WO disclosed