SCHEMBL7755948

SCHEMBL7755948

COC(CNc1ccccc1)CN1CCN(CCCC(c2ccc(F)cc2)c2ccc(F)cc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 8/20 0.52
SLC6A4 P31645 5/20 0.52
CYP3A4 P08684 4/20 0.48
CYP2D6 P10635 4/20 0.48
MAPK1 P28482 3/20 0.48
MTOR P42345 3/20 0.48
RAB9A P51151 3/20 0.48
TSHR P16473 2/20 0.48
FAAH O00519 1/20 0.48
ALOX12 P18054 1/20 0.48
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
BLM P54132 2/20 0.47
PMP22 Q01453 2/20 0.47
KCNH2 Q12809 6/20 0.47
HTR2A P28223 5/20 0.47
ADRA1A P35348 5/20 0.47
HRH1 P35367 5/20 0.47
DRD3 P35462 5/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7545277 0.99 SLC6A3 (0.51) SLC6A3SLC6A4CYP3A4CYP2D6MAPK1
SCHEMBL7757442 0.87 CYP3A4 (0.52) SLC6A3SLC6A4CYP3A4CYP2D6MAPK1
SCHEMBL4760958 0.84 CYP3A4 (0.51) SLC6A3SLC6A4CYP3A4CYP2D6MAPK1
SCHEMBL8615736 0.84 CYP3A4 (0.51) SLC6A3SLC6A4CYP3A4CYP2D6MAPK1
SCHEMBL8616378 0.84 CYP3A4 (0.51) SLC6A3SLC6A4CYP3A4CYP2D6MAPK1
Maleic Acid SCHEMBL8650751 0.83 CYP3A4 (0.48) SLC6A3SLC6A4CYP3A4CYP2D6MAPK1
Hydrochloric Acid SCHEMBL7543578 0.83 MEN1 (0.52) SLC6A3SLC6A4CYP3A4CYP2D6MAPK1
Hydrochloric Acid SCHEMBL8867248 0.83 MEN1 (0.52) SLC6A3SLC6A4CYP3A4CYP2D6MAPK1
Difluanine SCHEMBL1813120 0.81 SCN5A (0.59) SLC6A3SLC6A4CYP3A4CYP2D6MAPK1
SCHEMBL8614994 0.81 SLC6A3 (0.52) SLC6A3SLC6A4CYP3A4CYP2D6MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0706796-B1 DOPAMINE RE-UPTAKE INHIBITORS FOR THE TREATMENT OF PARKINSON'S SYNDROME POLA CHEM IND INC (JP) 2001-02-28 EP claimed
US-5747493-A N-/DIPHENYLALKYL/-PIPERAZINYL-2-HYDROXYPROPYLAMINES POLA CHEMICAL INDUSTRIES, INC. (JP) 1998-05-05 US claimed
EP-0706796-A1 DOPAMINE REINCORPORATION INHIBITOR POLA CHEMICAL INDUSTRIES, INC. (JP) 1996-04-17 EP claimed