SCHEMBL7763378

SCHEMBL7763378

NS(=O)(=O)N1CCN(CC(=O)O)CC1

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.47
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
ALDH1A1 P00352 2/20 0.39
SLC6A9 P48067 1/20 0.38
CHRNB2 P17787 3/20 0.37
CHRNB4 P30926 3/20 0.37
CHRNA3 P32297 3/20 0.37
CHRNA4 P43681 3/20 0.37
KMT2A Q03164 1/20 0.34
S1PR1 P21453 1/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7764777 0.83 ALDH1A1 (0.54) CA1CA2ALDH1A1CHRNB2CHRNB4
SCHEMBL7764241 0.81 CA1 (0.39) CA1CA2ALDH1A1CHRNB2CHRNB4
SCHEMBL3668924 0.81 MAPT (0.46) HSD17B10ALDH1A1KDM4E
SCHEMBL8742068 0.81 MAPT (0.46) HSD17B10ALDH1A1KDM4E
SCHEMBL16879998 0.81 KDM4E (0.47) HSD17B10ALDH1A1KMT2AKDM4E
Tetraxetan SCHEMBL18018 0.81 HSD17B10 (0.64) HSD17B10ALDH1A1SLC6A9S1PR1KDM4E
Tetraxetan SCHEMBL2635294 0.81 HSD17B10 (0.64) HSD17B10ALDH1A1SLC6A9S1PR1KDM4E
SCHEMBL6848102 0.81 HSD17B10 (0.64) HSD17B10ALDH1A1SLC6A9S1PR1KDM4E
SCHEMBL321989 0.81 HSD17B10 (0.64) HSD17B10ALDH1A1SLC6A9S1PR1KDM4E
Tetraxetan SCHEMBL2017956 0.81 HSD17B10 (0.64) HSD17B10ALDH1A1SLC6A9S1PR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1102789-A1 MONOCYCLIC COMPOUNDS HAVING NK-2 ANTAGONIST ACTION AND COMPOSITIONS CONTAINING THEM Menarini Ricerche S.p.A. (IT) 2001-05-30 EP disclosed
WO-2000008046-A1 MONOCYCLIC COMPOUNDS HAVING NK-2 ANTAGONIST ACTION AND COMPOSITIONS CONTAINING THEM MENARINI RICERCHE S.P.A. (IT) 2000-02-17 WO disclosed