SCHEMBL7765065

SCHEMBL7765065

Clc1ccc(Nc2ncccn2)cc1Cl

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.55
HDAC1 Q13547 1/20 0.55
HDAC2 Q92769 1/20 0.55
HDAC6 Q9UBN7 1/20 0.55
GRM4 Q14833 2/20 0.53
NPSR1 Q6W5P4 1/20 0.53
CDK4 P11802 1/20 0.49
CDK2 P24941 1/20 0.49
GSK3B P49841 1/20 0.49
KDR P35968 1/20 0.49
NPY5R Q15761 1/20 0.49
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
RAB9A P51151 2/20 0.47
NPC1 O15118 1/20 0.47
POLA1 P09884 2/20 0.47
IDO1 P14902 1/20 0.47
TDO2 P48775 1/20 0.47
RAPGEF4 Q8WZA2 1/20 0.46
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3034640 0.83 BRAF (0.52) HDAC3HDAC1HDAC2HDAC6GRM4
SCHEMBL14800759 0.80 HDAC3 (0.56) HDAC3HDAC1HDAC2HDAC6CDK4
SCHEMBL7981759 0.79 KMT2A (0.63) GRM4NPSR1KDRMEN1KMT2A
SCHEMBL31220846 0.79 KMT2A (0.63) GRM4NPSR1KDRMEN1KMT2A
SCHEMBL3584937 0.79 HDAC3 (0.63) HDAC3HDAC1HDAC2HDAC6CDK4
SCHEMBL12483125 0.78 POLB (0.57) HDAC3HDAC1HDAC2HDAC6CDK2
SCHEMBL12614443 0.78 RAPGEF4 (0.59) HDAC3HDAC1HDAC2HDAC6MEN1
SCHEMBL27714382 0.77 SCN9A (0.59) HDAC3HDAC1HDAC2HDAC6CDK2
SCHEMBL3951245 0.76 HDAC6 (0.58) HDAC3HDAC1HDAC2HDAC6GRM4
SCHEMBL8973728 0.76 NFKB1 (0.57) HDAC3HDAC1HDAC2HDAC6NPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1107957-A1 PYRIMIDINE COMPOUNDS AstraZeneca AB (SE) 2001-06-20 EP claimed
WO-2000012485-A1 PYRIMIDINE COMPOUNDS ASTRAZENECA AB (SE) 2000-03-09 WO claimed