SCHEMBL7765077

SCHEMBL7765077

CC(C)CN(c1cccc(CC(C)CNC(=O)[C@@H](C)CS(C)(=O)=O)c1O)S(=O)(=O)c1ccc2c(c1)OCCO2

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 2/20 0.41
MMP13 P45452 2/20 0.41
GAA P10253 2/20 0.40
HPGD P15428 1/20 0.40
KEAP1 Q14145 2/20 0.40
NFE2L2 Q16236 2/20 0.40
ALDH1A1 P00352 3/20 0.38
NPSR1 Q6W5P4 2/20 0.38
POLB P06746 1/20 0.38
RORC P51449 3/20 0.37
LMNA P02545 2/20 0.36
HTT P42858 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
RAB9A P51151 1/20 0.36
USP2 O75604 1/20 0.35
MAPT P10636 1/20 0.35
NPC1 O15118 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5689205 0.97 KEAP1 (0.40) MMP2MMP13GAAHPGDKEAP1
SCHEMBL7956674 0.88 KEAP1 (0.40) MMP2MMP13GAAHPGDKEAP1
SCHEMBL7955245 0.88 KEAP1 (0.40) MMP2MMP13GAAHPGDKEAP1
SCHEMBL7953042 0.86 KEAP1 (0.39) MMP2MMP13GAAHPGDKEAP1
SCHEMBL7959894 0.85 KEAP1 (0.38) MMP2MMP13GAAHPGDKEAP1
SCHEMBL5691126 0.84 KEAP1 (0.39) MMP2MMP13GAAHPGDKEAP1
Hydrochloric Acid SCHEMBL5506705 0.82 KEAP1 (0.38) MMP2MMP13GAAHPGDKEAP1
SCHEMBL5928160 0.82 KEAP1 (0.38) MMP2MMP13GAAHPGDKEAP1
SCHEMBL7945958 0.82 RORC (0.35) RORC
SCHEMBL6101123 0.81 CYP3A4 (0.37) HPGDALDH1A1RORCLMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0813519-B1 SULFONYLALKANOYLAMINO HYDROXYETHYLAMINO SULFONAMIDE RETROVIRAL PROTEASE INHIBITORS SEARLE & CO (US) 2001-05-09 EP disclosed
US-6169085-B1 A VIRICIDE FOR PREVENTING AND TREATING RETROVIRAL INFECTION OR THE SPREAD OF A RETROVIRUS, INHIBITING REPLICATION OF A RETROVIRUS AND TREATING AIDS G. D. SEARLE & COMPANY 2001-01-02 US disclosed
EP-1052250-A1 Sulfonylalkanoylamino hydroxyethylamino sulfonamide retroviral protease inhibitors G.D. SEARLE & CO. (US) 2000-11-15 EP disclosed