SCHEMBL7765521

SCHEMBL7765521

COc1ccc(N2CCN(Cc3ccc4c(c3)oc(=O)n4C)CC2)cc1

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 4/20 0.67
ALDH1A1 P00352 5/20 0.62
TSHR P16473 1/20 0.62
MAPK1 P28482 1/20 0.62
DRD3 P35462 1/20 0.55
DRD2 P14416 2/20 0.54
HTR1A P08908 2/20 0.53
SLC6A2 P23975 1/20 0.52
SLC6A4 P31645 1/20 0.52
SLC6A3 Q01959 1/20 0.52
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
USP2 O75604 2/20 0.48
KDM4E B2RXH2 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
CA12 O43570 1/20 0.48
CA9 Q16790 1/20 0.48
MAPT P10636 2/20 0.48
NPSR1 Q6W5P4 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7765509 0.89 MEN1 (0.64) DRD4ALDH1A1TSHRMAPK1DRD2
SCHEMBL7765531 0.87 DRD4 (0.64) DRD4ALDH1A1MAPK1DRD3DRD2
SCHEMBL7765547 0.83 USP2 (0.56) DRD4ALDH1A1TSHRMAPK1DRD2
SCHEMBL7766439 0.81 HTR1A (0.79) DRD4ALDH1A1MAPK1DRD3DRD2
Hydrochloric Acid SCHEMBL8403761 0.80 HTR1A (0.77) DRD4ALDH1A1MAPK1DRD3DRD2
SCHEMBL7767373 0.78 HTR1A (0.62) DRD4ALDH1A1DRD3DRD2HTR1A
SCHEMBL7762726 0.77 MEN1 (0.62) DRD4ALDH1A1DRD2HTR1AMEN1
SCHEMBL10982732 0.77 HTR1A (0.66) DRD4ALDH1A1TSHRMAPK1HTR1A
Hydrochloric Acid SCHEMBL8403646 0.76 MEN1 (0.61) DRD4ALDH1A1DRD2HTR1AMEN1
SCHEMBL10392906 0.75 HTR1A (0.62) DRD4ALDH1A1TSHRMAPK1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1072655-C New heterocyclic aminomethyl compounds, process for preparing them and pharmaceutical compositions containing them ADIR (FR) 2001-10-10 CN claimed
EP-0841330-B1 Aminomethyl heterocyclic derivatives, process of their preparation and pharmaceutical compositions containing them ADIR (FR) 2001-06-27 EP claimed
CN-1182083-A New heterocyclic aminomethyl compounds, process for preparing them and pharmaceutical compositions containing them ADIR (FR) 1998-05-20 CN claimed
EP-0841330-A1 Aminomethyl heterocyclic derivatives, process of their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1998-05-13 EP claimed
CN-1072655-C New heterocyclic aminomethyl compounds, process for preparing them and pharmaceutical compositions containing them ADIR (FR) 2001-10-10 CN disclosed
EP-0841330-B1 Aminomethyl heterocyclic derivatives, process of their preparation and pharmaceutical compositions containing them ADIR (FR) 2001-06-27 EP disclosed
US-5919784-A ANXIETY, DEPRESSION ADIR ET COMPAGNIE (FR) 1999-07-06 US disclosed
CN-1182083-A New heterocyclic aminomethyl compounds, process for preparing them and pharmaceutical compositions containing them ADIR (FR) 1998-05-20 CN disclosed
EP-0841330-A1 Aminomethyl heterocyclic derivatives, process of their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1998-05-13 EP disclosed