SCHEMBL7765792

SCHEMBL7765792

CCCC(=O)[N]NC(=O)C(Cl)Cl

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.34
ALDH1A2 O94788 1/20 0.33
ALDH1A1 P00352 1/20 0.33
ALDH2 P05091 1/20 0.33
ALDH1A3 P47895 1/20 0.33
HDAC3 O15379 3/20 0.32
HDAC1 Q13547 3/20 0.32
HDAC2 Q92769 3/20 0.32
HDAC8 Q9BY41 3/20 0.32
HDAC6 Q9UBN7 1/20 0.32
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32
CTSD P07339 1/20 0.31
FFAR3 O14843 2/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7771405 0.89 ALDH1A1 (0.39) TSHRALDH1A2ALDH1A1ALDH2ALDH1A3
SCHEMBL7773745 0.83 ALDH1A2 (0.35) ALDH1A2ALDH1A1ALDH2ALDH1A3CYP3A4
SCHEMBL7771071 0.80 CES2 (0.35) TSHRHDAC3HDAC1HDAC2HDAC8
SCHEMBL9821272 0.74 CES1 (0.38) TSHRALDH1A1HDAC3HDAC1HDAC2
SCHEMBL8822944 0.73 HDAC3 (0.38) TSHRALDH1A1HDAC3HDAC1HDAC2
SCHEMBL7771366 0.72 TSHR (0.34) TSHRHDAC3HDAC1HDAC2HDAC8
SCHEMBL7765741 0.72 ALDH1A2 (0.34) ALDH1A2ALDH1A1ALDH2ALDH1A3
SCHEMBL7770074 0.71 HDAC3 (0.39) TSHRALDH1A1HDAC3HDAC1HDAC2
SCHEMBL7769331 0.69 HDAC3 (0.38) TSHRALDH1A1HDAC3HDAC1HDAC2
SCHEMBL7769432 0.69 HDAC3 (0.38) TSHRALDH1A1HDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0765879-B1 13-Substituted milbemycin 5-oxime derivatives, their preparation and their use against insects and other pests SANKYO CO (JP) 2001-02-14 EP disclosed
US-5861429-A MITICIDES AND ANTHELMINTICS SANKYO COMPANY, LIMITED (JP) 1999-01-19 US disclosed
EP-0765879-A1 13-Substituted milbemycin 5-oxime derivatives, their preparation and their use against insects and other pests SANKYO COMPANY LIMITED (JP) 1997-04-02 EP disclosed