SCHEMBL7765980

SCHEMBL7765980

CCCCC(=O)[N]NC(=O)C(F)F

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CES2 O00748 5/20 0.41
CES1 P23141 5/20 0.37
ALDH1A1 P00352 2/20 0.34
TP53 P04637 1/20 0.34
CA1 P00915 3/20 0.33
MAPT P10636 1/20 0.32
CA2 P00918 2/20 0.32
FAAH O00519 2/20 0.32
MEN1 O00255 1/20 0.32
MAPK1 P28482 1/20 0.32
KMT2A Q03164 1/20 0.32
RAB9A P51151 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
HSP90AA1 P07900 1/20 0.31
NPSR1 Q6W5P4 1/20 0.30
AKR1B1 P15121 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7771071 0.89 CES2 (0.35) CES2CES1
SCHEMBL7771405 0.81 ALDH1A1 (0.39) CES2CES1ALDH1A1TP53CA1
SCHEMBL7773730 0.80
SCHEMBL7771427 0.76 CES1 (0.38) CES2CES1ALDH1A1TP53CA1
SCHEMBL7769364 0.74 EPHX1 (0.46) CES2CES1ALDH1A1FAAHMEN1
SCHEMBL7770041 0.73 CES1 (0.39) CES2CES1ALDH1A1TP53CA1
SCHEMBL7769860 0.73 ALDH1A1 (0.40) CES2CES1ALDH1A1MAPTFAAH
SCHEMBL7769447 0.72 FAAH (0.42) CES2CES1ALDH1A1TP53CA1
SCHEMBL7766040 0.72 CES1 (0.38) CES2CES1ALDH1A1TP53CA1
SCHEMBL7771382 0.71 ALDH1A1 (0.42) ALDH1A1MAPTFAAHMEN1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0765879-B1 13-Substituted milbemycin 5-oxime derivatives, their preparation and their use against insects and other pests SANKYO CO (JP) 2001-02-14 EP disclosed
EP-0765879-A1 13-Substituted milbemycin 5-oxime derivatives, their preparation and their use against insects and other pests SANKYO COMPANY LIMITED (JP) 1997-04-02 EP disclosed